SCHEMBL4255348

SCHEMBL4255348

CCCCCCCCCOC(=O)C(F)(F)F

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CES2 O00748 4/20 0.58
NAAA Q02083 1/20 0.55
EPHX1 P07099 1/20 0.52
FAAH O00519 8/20 0.50
CES1 P23141 5/20 0.50
TSHR P16473 2/20 0.50
MEN1 O00255 1/20 0.50
CYP1A2 P05177 1/20 0.50
KMT2A Q03164 1/20 0.50
HSD17B10 Q99714 1/20 0.50
HCAR2 Q8TDS4 1/20 0.47
RAD52 P43351 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5470496 1.00 CES2 (0.58) CES2NAAAEPHX1FAAHCES1
SCHEMBL4765360 1.00 CES2 (0.58) CES2NAAAEPHX1FAAHCES1
SCHEMBL28781368 1.00 CES2 (0.58) CES2NAAAEPHX1FAAHCES1
SCHEMBL28472787 1.00 CES2 (0.58) CES2NAAAEPHX1FAAHCES1
SCHEMBL4361492 1.00 CES2 (0.58) CES2NAAAEPHX1FAAHCES1
SCHEMBL1123659 1.00 CES2 (0.58) CES2NAAAEPHX1FAAHCES1
SCHEMBL4080844 1.00 CES2 (0.58) CES2NAAAEPHX1FAAHCES1
SCHEMBL30475134 1.00 CES2 (0.58) CES2NAAAEPHX1FAAHCES1
SCHEMBL2691990 1.00 CES2 (0.58) CES2NAAAEPHX1FAAHCES1
SCHEMBL2691404 1.00 CES2 (0.58) CES2NAAAEPHX1FAAHCES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 49 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116284233-B Method for preparing itracin 浙江湃肽生物股份有限公司 2024-07-05 CN disclosed
CN-118255772-A Quinazoline derivatives as antitumor agents 苏州赞荣医药科技有限公司 2024-06-28 CN disclosed
CN-114728938-B Tetrahydroisoquinoline spiro compounds as PRMT5 inhibitors 南京再明医药有限公司 2024-05-24 CN disclosed
CN-117858872-A Heterocyclic EGFR inhibitors for the treatment of cancer 缆图药品公司 2024-04-09 CN disclosed
CN-110637025-B Peptide amide compound, preparation method and medical application thereof 四川海思科制药有限公司 2023-07-18 CN disclosed
CN-116284233-A Method for preparing itracin 浙江湃肽生物股份有限公司 2023-06-23 CN disclosed
CN-115996912-A Iminothiolanone inhibitors of ENPP1 沃拉斯查疗法公司 2023-04-21 CN disclosed
CN-114728938-A Tetrahydroisoquinoline spiro compounds as PRMT5 inhibitors 江苏先声药业有限公司 2022-07-08 CN disclosed
CN-114364682-A Compound 4,4A,5,7,8, 8A-hexapyrido [4,3-B ] [1,4] oxazin-3-one as MAGL inhibitor 豪夫迈·罗氏有限公司 2022-04-15 CN disclosed
CN-114364684-A Heterocyclic compounds 豪夫迈·罗氏有限公司 2022-04-15 CN disclosed
CN-101501006-A Pyridone and pyridazinone derivatives as poly (ADP-ribose) polymerase (PARP) inhibitors ANGELETTI P IST RICHERCHE BIO (IT) 2009-08-05 CN disclosed
CN-101448825-A CNS active fused bicyclic heterocycle substituted azabicycloalkane derivatives ABBOTT LAB (US) 2009-06-03 CN disclosed
CN-101291931-A 9-azabicyclo [3.3.1]nonane derivatives as monoamine reuptake inhibitors ORGANON NV (NL) 2008-10-22 CN disclosed
WO-2008057938-A1 NICOTINIC ACETYLCHOLINE RECEPTORSUB-TYPE SELECTIVE AMIDES OF DIAZABICYCLOALKANES TARGACEPT, INC. (US) 2008-05-15 WO disclosed
CN-1898239-A Novel diazaspiroalkanes and their use in the treatment of CCR8 mediated diseases ASTRAZENECA AB (SE) 2007-01-17 CN disclosed
EP-1626970-A1 AZABICYCLOALKANE COMPOUNDS AS MUSCARINIC RECEPTOR ANTAGONISTS Theravance, Inc. (US) 2006-02-22 EP disclosed
WO-2004106333-A1 AZABICYCLOALKANE COMPOUNDS AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE, INC. (US) 2004-12-09 WO disclosed
CN-1449408-A Synthetic methods for Aplidine and novel antitumor derivatives, and methods of making and using the same PHARMA MAR SA (ES) 2003-10-15 CN disclosed
US-5466877-A Fluorination with deesterification and alkylation MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1995-11-14 US disclosed
WO-1995025082-A1 PROCESS FOR CONVERTING PERFLUORINATED ESTERS TO PERFLUORINATED ACYL FLUORIDES AND/OR KETONES MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1995-09-21 WO disclosed