SCHEMBL4257425

SCHEMBL4257425

CC(C)c1cc(C(=O)N2Cc3cccc(OC(C)(C)CN)c3C2)c(O)cc1O

nearest known ligand 0.60

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 16/20 0.60
HSP90AB1 P08238 15/20 0.60
HSP90B1 P14625 4/20 0.49
TRAP1 Q12931 2/20 0.49
HDAC8 Q9BY41 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL383083 0.79 HSP90AA1 (0.60) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL383810 0.79 HSP90AA1 (0.59) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL10214759 0.78 HSP90AB1 (0.73) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL19339155 0.77 HSP90AB1 (0.69) HSP90AA1HSP90AB1HSP90B1
SCHEMBL30091904 0.77 HSP90AB1 (1.00) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL383624 0.77 HSP90AB1 (1.00) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL30091906 0.77 HSP90AB1 (1.00) HSP90AA1HSP90AB1HSP90B1TRAP1
Hydrochloric Acid SCHEMBL382762 0.77 HSP90AB1 (0.72) HSP90AA1HSP90AB1HSP90B1TRAP1
SCHEMBL19339221 0.76 HSP90AA1 (0.56) HSP90AA1HSP90AB1HSP90B1TRAP1HDAC8
Hypochlorous Acid SCHEMBL12802787 0.76 HSP90AB1 (0.70) HSP90AA1HSP90AB1HSP90B1TRAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2081891-A2 PHARMACEUTICAL COMPOUNDS HAVING HSP90 INHIBITORY OR MODULATING ACTIVITY Astex Therapeutics Limited (GB) 2009-07-29 EP disclosed
WO-2008044027-A2 PHARMACEUTICAL COMPOUNDS HAVING HSP90 INHIBITORY OR MODULATING ACTIVITY ASTEX THERAPEUTICS LIMITED (GB) 2008-04-17 WO disclosed