SCHEMBL4257537

SCHEMBL4257537

C=CCC(C(=O)NC)c1ccc(F)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.46
FFAR2 O15552 1/20 0.42
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC10 Q969S8 1/20 0.41
HDAC11 Q96DB2 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
HDAC9 Q9UKV0 1/20 0.41
HDAC5 Q9UQL6 1/20 0.41
TGM2 P21980 1/20 0.40
HTT P42858 1/20 0.38
KCNQ2 O43526 1/20 0.36
POLB P06746 1/20 0.36
MME P08473 1/20 0.36
LMNA P02545 1/20 0.36
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6002600 0.85 CYP2C19 (0.44) CYP2C19FFAR2HDAC3HDAC4HDAC1
SCHEMBL4262027 0.85 CYP2C19 (0.44) CYP2C19FFAR2HDAC3HDAC4HDAC1
SCHEMBL9114406 0.84 CYP2C19 (0.67) CYP2C19FFAR2HDAC3HDAC4HDAC1
SCHEMBL960592 0.80 CYP2C19 (0.71) CYP2C19FFAR2HDAC3HDAC4HDAC1
SCHEMBL4265668 0.80 CYP2C19 (0.71) CYP2C19FFAR2HDAC3HDAC4HDAC1
SCHEMBL4264360 0.79 CYP2C19 (0.50) CYP2C19FFAR2HDAC3HDAC4HDAC1
SCHEMBL6002239 0.79 CYP2C19 (0.50) CYP2C19FFAR2HDAC3HDAC4HDAC1
SCHEMBL9045383 0.78 ALDH1A1 (0.43) CYP2C19FFAR2HTTKCNQ2LMNA
SCHEMBL20993324 0.76 CNR1 (0.44) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL28608516 0.74 CYP2C19 (0.57) CYP2C19HTTLMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1636221-B1 3-Heterocyclyl-Azetidine compounds useful as NK1/NK2 receptors antagonists ALBIREO AB (SE) 2009-08-12 EP disclosed
US-20090023731-A1 SOLUBLE EPOXIDE HYDROLASE INHIBITORS ARETE THERAPEUTICS, INC. 2009-01-22 US disclosed
WO-2008116145-A2 SOLUBLE EPOXIDE HYDROLASE INHIBITORS ARETE THERAPEUTICS, INC. (US) 2008-09-25 WO disclosed
US-7402581-B2 Azetidine compounds ALBIREO AB (SE) 2008-07-22 US disclosed
US-20060172988-A1 Azetidine compounds ALBIREO AB (SE) 2006-08-03 US disclosed
EP-1636221-A2 NEW AZETIDINE COMPOUNDS AstraZeneca AB (SE) 2006-03-22 EP disclosed
WO-2004110344-A2 NEW AZETIDINE COMPOUNDS ASTRAZENECA AB (SE) 2004-12-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090023731-A1 SOLUBLE EPOXIDE HYDROLASE INHIBITORS EPHX1, EPHX2, NCEH1 CYP2C19 912/4885FFAR2 812/4885HDAC3 4415/4885
US-20060172988-A1 Azetidine compounds HRH2, HRH4, HRH1 CYP2C19 9/4885FFAR2 2459/4885HDAC3 1747/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.