SCHEMBL4257664

SCHEMBL4257664

CCN(CC)CC.NC(=O)c1cnc[nH]1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AOC1 P19801 1/20 0.43
HRH3 Q9Y5N1 6/20 0.41
HRH4 Q9H3N8 5/20 0.41
GAA P10253 1/20 0.40
ESR1 P03372 2/20 0.39
CYP19A1 P11511 2/20 0.39
TP53 P04637 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
ALDH1A1 P00352 2/20 0.37
CYP3A4 P08684 2/20 0.37
GABRA1 P14867 1/20 0.37
TSHR P16473 1/20 0.37
NFKB1 P19838 1/20 0.37
GABRR1 P24046 1/20 0.37
GABRR2 P28476 1/20 0.37
GABRA5 P31644 1/20 0.37
GABRB2 P47870 1/20 0.37
GABRA4 P48169 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL826324 0.85
Hydrochloric Acid SCHEMBL17843027 0.83
Bromide SCHEMBL28268955 0.83 AOC1 (0.48) AOC1HRH3GAAESR1CYP19A1
Hydrochloric Acid SCHEMBL2452413 0.83 AOC1 (0.48) AOC1HRH3GAAESR1CYP19A1
Water SCHEMBL27319944 0.83
Hydrochloric Acid SCHEMBL29686657 0.83 AOC1 (0.48) AOC1HRH3GAAESR1CYP19A1
Formic Acid SCHEMBL23930802 0.78 AOC1 (0.44) AOC1HRH3GAAESR1CYP19A1
Trifluoroacetic Acid SCHEMBL3635857 0.75 HRH3 (0.54) AOC1HRH3HRH4GAATP53
SCHEMBL8546519 0.75 AOC1 (0.42) AOC1HRH3GAAESR1CYP19A1
SCHEMBL16950288 0.74 AOC1 (0.41) AOC1HRH3HRH4GAAESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010535-A1 THIOXANTHINE DERIVATIVES AND THEIR USE AS INHIBITORS OF MPO AstraZeneca AB (SE) 2009-01-07 EP disclosed
WO-2007120098-A1 THIOXANTHINE DERIVATIVES AND THEIR USE AS INHIBITORS OF MPO ASTRAZENECA AB (SE) 2007-10-25 WO disclosed