SCHEMBL4258306

SCHEMBL4258306

CC1=C(C(=O)O)C(c2ccccc2-c2ccc(C(C)O)cc2)n2nnnc2N1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.51
LMNA P02545 3/20 0.49
KMT2A Q03164 2/20 0.48
HTT P42858 1/20 0.48
SMN1; SMN2 Q16637 3/20 0.47
MAPT P10636 2/20 0.47
TP53 P04637 1/20 0.47
THRB P10828 1/20 0.46
GAA P10253 1/20 0.46
NPSR1 Q6W5P4 2/20 0.45
PKM P14618 1/20 0.44
POLB P06746 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2996994 0.86 ALDH1A1 (0.60) ALDH1A1LMNAKMT2AHTTSMN1; SMN2
SCHEMBL3005370 0.85 KMT2A (0.54) ALDH1A1LMNAKMT2AHTTSMN1; SMN2
SCHEMBL2992365 0.84 ALDH1A1 (0.51) ALDH1A1LMNAKMT2AHTTSMN1; SMN2
SCHEMBL3003897 0.81 ALDH1A1 (0.52) ALDH1A1LMNAKMT2AHTTSMN1; SMN2
SCHEMBL3250826 0.79 ALDH1A1 (0.58) ALDH1A1LMNAKMT2AHTTSMN1; SMN2
SCHEMBL3004302 0.78 KMT2A (0.52) ALDH1A1LMNAKMT2AHTTSMN1; SMN2
SCHEMBL3000251 0.78 ALDH1A1 (0.48) ALDH1A1LMNAKMT2AHTTSMN1; SMN2
SCHEMBL2993898 0.76 ALDH1A1 (0.56) ALDH1A1LMNAKMT2AHTTSMN1; SMN2
SCHEMBL3002840 0.76 ALDH1A1 (0.63) ALDH1A1LMNAKMT2AHTTSMN1; SMN2
SCHEMBL3246503 0.75 ALDH1A1 (0.68) ALDH1A1LMNAKMT2AHTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009006580-A1 OPTIONALLY CONDENSED DIHYDROPYRIDINE, DIHYDROPYRIMIDINE AND DIHYDROPYRANE DERIVATIVES ACTING AS LATE SODIUM CHANNEL BLOCKERS CV THERAPEUTICS, INC. (US) 2009-01-08 WO disclosed