SCHEMBL4258455

SCHEMBL4258455

COc1cc(C=O)ccc1Oc1ccc(N)cc1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTR P02766 1/20 0.72
ALDH1A1 P00352 8/20 0.64
TSHR P16473 1/20 0.64
CYP19A1 P11511 4/20 0.57
FDPS P14324 1/20 0.55
HPGD P15428 2/20 0.54
TRIM24 O15164 1/20 0.54
ALDH5A1 P51649 1/20 0.54
ABAT P80404 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
TRIM33 Q9UPN9 1/20 0.54
MAPT P10636 3/20 0.51
AOX1 Q06278 1/20 0.50
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
NQO2 P16083 1/20 0.47
ALDH1A3 P47895 1/20 0.47
TUBB4A P04350 1/20 0.46
TUBB P07437 1/20 0.46
TUBA3C P0DPH7 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17955067 0.90 TTR (0.81) TTRALDH1A1TSHRFDPSHPGD
SCHEMBL26936583 0.89 TTR (0.79) TTRALDH1A1TSHRFDPSHPGD
SCHEMBL27670275 0.86 TTR (0.74) TTRALDH1A1TSHRFDPSHPGD
SCHEMBL26936729 0.84 TTR (0.72) TTRALDH1A1TSHRFDPSHPGD
SCHEMBL26936448 0.84 TTR (0.72) TTRALDH1A1TSHRFDPSHPGD
SCHEMBL27983148 0.84 TTR (0.72) TTRALDH1A1TSHRFDPSHPGD
SCHEMBL1616189 0.84 TTR (1.00) TTRALDH1A1TSHRFDPSHPGD
SCHEMBL31238528 0.84 TTR (1.00) TTRALDH1A1TSHRFDPSHPGD
SCHEMBL1869030 0.83 ALDH1A1 (0.84) TTRALDH1A1TSHRFDPSHPGD
SCHEMBL17508149 0.82 TTR (0.69) TTRALDH1A1TSHRFDPSHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2450352-A1 PROPHYLACTIC OR THERAPEUTIC AGENT FOR CANCER Takeda Pharmaceutical Company Limited (JP) 2012-05-09 EP disclosed
WO-2011016501-A1 PROPHYLACTIC OR THERAPEUTIC AGENT FOR CANCER 武田薬品工業株式会社 (JP) 2011-02-10 WO disclosed