Cortodoxone

Cortodoxone

SCHEMBL42590

C[C@]12CCC(=O)C=C1CC[C@@H]1[C@@H]2CC[C@@]2(C)[C@H]1CC[C@]2(O)C(=O)CO

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 8/20 1.00
SHBG P04278 7/20 1.00
SMN1; SMN2 Q16637 7/20 1.00
SERPINA6 P08185 6/20 1.00
CYP2C19 P33261 5/20 1.00
HIF1A Q16665 5/20 1.00
LMNA P02545 5/20 1.00
CYP3A4 P08684 4/20 1.00
TSHR P16473 3/20 1.00
BLM P54132 2/20 1.00
PMP22 Q01453 2/20 1.00
NR3C1 P04150 6/20 0.78
KMT2A Q03164 3/20 0.78
MAPT P10636 3/20 0.78
MEN1 O00255 2/20 0.78
ADORA3 P0DMS8 1/20 0.78
MAPK3 P27361 1/20 0.78
SLC6A3 Q01959 1/20 0.78
ALDH1A1 P00352 4/20 0.74
CYP2D6 P10635 1/20 0.74

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cortodoxone SCHEMBL16834876 1.00 HSD17B10 (1.00) HSD17B10SHBGSMN1; SMN2SERPINA6CYP2C19
Cortodoxone SCHEMBL3641463 1.00 HSD17B10 (1.00) HSD17B10SHBGSMN1; SMN2SERPINA6CYP2C19
Cortodoxone SCHEMBL1592553 1.00 HSD17B10 (1.00) HSD17B10SHBGSMN1; SMN2SERPINA6CYP2C19
Cortodoxone SCHEMBL13352414 1.00 HSD17B10 (1.00) HSD17B10SHBGSMN1; SMN2SERPINA6CYP2C19
Cortodoxone SCHEMBL1592718 1.00 HSD17B10 (1.00) HSD17B10SHBGSMN1; SMN2SERPINA6CYP2C19
Cortodoxone SCHEMBL24900239 1.00 HSD17B10 (1.00) HSD17B10SHBGSMN1; SMN2SERPINA6CYP2C19
Cortodoxone SCHEMBL14360590 1.00 HSD17B10 (1.00) HSD17B10SHBGSMN1; SMN2SERPINA6CYP2C19
Cortodoxone SCHEMBL17906542 1.00 HSD17B10 (1.00) HSD17B10SHBGSMN1; SMN2SERPINA6CYP2C19
Cortodoxone SCHEMBL13768127 1.00 HSD17B10 (1.00) HSD17B10SHBGSMN1; SMN2SERPINA6CYP2C19
SCHEMBL6019058 0.91 HSD17B10 (0.84) HSD17B10SHBGSMN1; SMN2SERPINA6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 11710 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260148848-A1 BIOMARKERS FOR DIAGNOSIS AND TREATMENT OF ENDOCRINE HYPERTENSION, AND METHODS OF IDENTIFICATION THEREOF INSERM (INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE) (FR) 2026-05-28 US claimed
EP-4747627-A1 METHODS AND SYSTEMS FOR PREDICTIVE CLASSIFICATION BY MASS SPECTROMETRY AND TRAINED LARGE SPECTRAL MODELS Matterworks Inc (US) 2026-05-27 EP claimed
US-20260139030-A1 CHIMERIC PROTEINS FOR TREATING CUTANEOUS INFLAMMATION SHATTUCK LABS INC (US) 2026-05-21 US claimed
US-20260140124-A1 PCOS STRATIFICATION THE UNIVERSITY OF BIRMINGHAM (GB) 2026-05-21 US claimed
EP-4740024-A1 ENDOMETRIOSIS MARKERS AND METHODS OF DIAGNOSING ENDOMETRIOSIS The University Court Of The University of Edinburgh (GB) 2026-05-13 EP claimed
US-20260103492-A1 CYCLOSPORINE COMPOSITIONS AND METHODS OF USE BACAINN BIOTHERAPEUTICS, LTD. (KY) 2026-04-16 US claimed
EP-4718074-A2 MASS SPECTROMETRY ASSAY FOR CONGENITAL ADRENAL HYPERPLASIA Quest Diagnostics Investments Incorporated (US) 2026-04-01 EP claimed
EP-4718073-A2 MASS SPECTROMETRY ASSAY FOR CONGENITAL ADRENAL HYPERPLASIA Quest Diagnostics Investments Incorporated (US) 2026-04-01 EP claimed
EP-4687915-A1 CLASCOTERONE AND MINOXIDIL COMBINATION THERAPY FOR USE IN TREATING HAIR LOSS Cassiopea S.p.A. (IT) 2026-02-11 EP claimed
US-20250387412-A1 ENZYMATIC PROCESS FOR OBTAINING 17 ALPHA-MONOESTERS OF CORTEXOLONE AND/OR ITS 9,11-DEHYDRODERIVATIVES CASSIOPEA S.P.A. (IT) 2025-12-25 US claimed
EP-0218300-A2 Brain-specific drug delivery UNIVERSITY OF FLORIDA (US) 1987-04-15 EP claimed
EP-0186948-A1 Process and intermediates for the preparation of 17alpha-hydroxyprogesterones and corticoids from an enol steroid THE UPJOHN COMPANY (US) 1986-07-09 EP claimed
US-4540564-A DIHYDROPYRIDINE AND/OR PYRIDINIUM SALT REDOX CARRIER UNIVERSITY OF FLORIDA (US) 1985-09-10 US claimed
EP-0110955-A1 BRAIN-SPECIFIC DRUG DELIVERY. UNIV FLORIDA (US) 1984-06-20 EP claimed
WO-1983003968-A1 BRAIN-SPECIFIC DRUG DELIVERY UNIVERSITY OF FLORIDA (US) 1983-11-24 WO claimed
US-4391803-A STEROID BLEND HEPAR INDUSTRIES (US) 1983-07-05 US claimed
EP-0005476-B1 PROCESS FOR PREPARING HUMAN INTERFERON Dr. Karl Thomae GmbH (DE) 1981-12-30 EP claimed
US-4266024-A USING ALKYLENEDIAMIDES, DIMETHYL SULFOXIDE OR GLUCOCORTICOIDS AS STIMULATORS FOR LYMPHOID CELLS BOEHRINGER INGELHEIM GMBH (DE) 1981-05-05 US claimed
US-4220716-A Process for the preparation of 7α-hydroxylated steroids HOFFMANN-LA ROCHE INC. (US) 1980-09-02 US claimed
EP-0001102-A1 Process for the preparation of 7-hydroxy steroids F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1979-03-21 EP claimed