SCHEMBL4259616

SCHEMBL4259616

O=c1c(-c2ccccc2)c(O)nc2sc3ccccc3n12

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.62
CYP2C9 P11712 1/20 0.62
KDM4E B2RXH2 5/20 0.58
LMNA P02545 4/20 0.58
SMN1; SMN2 Q16637 3/20 0.58
RAB9A P51151 3/20 0.58
NPC1 O15118 2/20 0.58
HPGD P15428 2/20 0.58
TP53 P04637 1/20 0.58
HSD17B10 Q99714 1/20 0.58
L3MBTL1 Q9Y468 3/20 0.49
PDE1B Q01064 1/20 0.49
PDE3A Q14432 1/20 0.49
PDE11A Q9HCR9 1/20 0.49
MAPK1 P28482 1/20 0.46
MAPT P10636 3/20 0.45
ALDH1A1 P00352 2/20 0.45
HTT P42858 2/20 0.45
POLB P06746 2/20 0.45
APEX1 P27695 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4399923 0.83 KDM4E (0.58) CYP1A2CYP2C9KDM4ELMNASMN1; SMN2
SCHEMBL4401354 0.78 KDM4E (0.52) CYP1A2CYP2C9KDM4ELMNASMN1; SMN2
SCHEMBL10660178 0.75 MAPT (0.51) CYP1A2CYP2C9KDM4ELMNASMN1; SMN2
SCHEMBL12289816 0.74 KDM4E (1.00) CYP1A2CYP2C9KDM4ELMNASMN1; SMN2
SCHEMBL24513417 0.73 KDM4E (0.71) CYP1A2CYP2C9KDM4ELMNASMN1; SMN2
SCHEMBL24513420 0.73 KDM4E (0.71) CYP1A2CYP2C9KDM4ELMNASMN1; SMN2
SCHEMBL24513181 0.73 KDM4E (0.49) CYP1A2CYP2C9KDM4ELMNASMN1; SMN2
SCHEMBL23075994 0.72 PDE1B (0.56) CYP1A2CYP2C9KDM4ELMNASMN1; SMN2
SCHEMBL635537 0.72 KDM4E (0.48) CYP1A2CYP2C9KDM4ELMNASMN1; SMN2
SCHEMBL9543555 0.72 CYP1A2 (0.65) CYP1A2CYP2C9KDM4ELMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7488721-B2 Real time methylumbelliferone-based assay MCMASTER UNIVERSITY (CA) 2009-02-10 US disclosed
US-7488721-B2 Real time methylumbelliferone-based assay MCMASTER UNIVERSITY (CA) 2009-02-10 US disclosed
US-7488721-B2 Real time methylumbelliferone-based assay MCMASTER UNIVERSITY (CA) 2009-02-10 US disclosed
US-20060008862-A1 Real time methylumbelliferone-based assay THE HOSPITAL FOR SICK CHILDREN 2006-01-12 US disclosed