SCHEMBL9543555

SCHEMBL9543555

CCOC(=O)c1c(O)nc2sc3ccccc3n2c1=O

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.65
CYP2C9 P11712 1/20 0.65
KDM4E B2RXH2 10/20 0.56
MAPT P10636 4/20 0.48
ALDH1A1 P00352 3/20 0.48
HPGD P15428 5/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
NPC1 O15118 1/20 0.48
LMNA P02545 1/20 0.48
TP53 P04637 1/20 0.48
RAB9A P51151 1/20 0.48
HSD17B10 Q99714 1/20 0.48
L3MBTL1 Q9Y468 4/20 0.47
MEN1 O00255 3/20 0.47
POLB P06746 3/20 0.47
KMT2A Q03164 3/20 0.47
CTDSP1 Q9GZU7 2/20 0.47
TDP1 Q9NUW8 2/20 0.46
HCRTR1 O43613 1/20 0.46
THRB P10828 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9540922 0.85 KDM4E (0.53) CYP1A2CYP2C9KDM4EMAPTALDH1A1
SCHEMBL10463716 0.78 KDM4E (0.51) CYP1A2CYP2C9KDM4EMAPTALDH1A1
SCHEMBL7331553 0.73 KDM4E (0.51) CYP1A2CYP2C9KDM4EMAPTALDH1A1
SCHEMBL4259616 0.72 CYP1A2 (0.62) CYP1A2CYP2C9KDM4EMAPTALDH1A1
SCHEMBL10464594 0.71 KDM4E (0.47) CYP1A2CYP2C9KDM4EMAPTALDH1A1
SCHEMBL13317085 0.71 KDM4E (0.60) CYP1A2CYP2C9KDM4EMAPTALDH1A1
SCHEMBL1582219 0.70 MAPK1 (0.60) CYP1A2CYP2C9KDM4EMAPTALDH1A1
SCHEMBL2922603 0.70 GAA (0.53) CYP1A2KDM4EMAPTALDH1A1SMN1; SMN2
SCHEMBL31629507 0.70 KDM4E (0.43) CYP1A2CYP2C9KDM4EMAPTALDH1A1
SCHEMBL12254659 0.70 KDM4E (0.43) CYP1A2CYP2C9KDM4EMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-5039293-A None JP disclosed
JP-H0539293-A IMMUNOMODULATING AGENT AND THIAZOLOPYRIMIDINE DERIVATIVE KYOWA HAKKO KOGYO CO LTD 1993-02-19 JP disclosed