SCHEMBL4260740

SCHEMBL4260740

CC1CNCC(C)N1c1nc2c(C(=O)NC3CN4CCC3CC4)cccc2o1

nearest known ligand 0.82

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 16/20 0.82
KCNH2 Q12809 5/20 0.68
CYP2C19 P33261 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1061935 1.00 HTR3A (0.82) HTR3AKCNH2CYP2C19
SCHEMBL1061932 1.00 HTR3A (0.82) HTR3AKCNH2CYP2C19
Hydrochloric Acid SCHEMBL1058485 0.99 HTR3A (0.80) HTR3AKCNH2CYP2C19
Hydrochloric Acid SCHEMBL1058491 0.99 HTR3A (0.80) HTR3AKCNH2CYP2C19
Hydrochloric Acid SCHEMBL1058488 0.99 HTR3A (0.80) HTR3AKCNH2CYP2C19
SCHEMBL1005719 0.90 HTR3A (1.00) HTR3AKCNH2CYP2C19
Hydrochloric Acid SCHEMBL1005563 0.89 HTR3A (0.98) HTR3AKCNH2CYP2C19
SCHEMBL8214868 0.89 HTR3A (0.65) HTR3AKCNH2CYP2C19
Hydrochloric Acid SCHEMBL1005561 0.89 HTR3A (0.98) HTR3AKCNH2CYP2C19
SCHEMBL8222039 0.89 HTR3A (0.70) HTR3AKCNH2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2061460-A2 2-AMINOBENZOXAZOLE CARBOXAMIDES AS 5HT3 MODULATORS Albany Molecular Research, Inc. (US) 2009-05-27 EP disclosed
WO-2008019372-A2 2-AMINOBENZOXAZOLE CARBOXAMIDES AS 5HT3 MODULATORS ALBANY MOLECULAR RESEARCH, INC. (US) 2008-02-14 WO disclosed