SCHEMBL4261685

SCHEMBL4261685

C[C@H](Cc1cccc(CCC(=O)O)c1)NC[C@H](O)c1ccc(OCc2ccccc2)c(CO)c1

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 15/20 0.56
ADRB3 P13945 7/20 0.51
ADRB1 P08588 4/20 0.49
CYP2D6 P10635 2/20 0.49
ADRA1D P25100 1/20 0.49
ADRA1A P35348 1/20 0.49
ADRA1B P35368 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
CYP3A4 P08684 1/20 0.47
HIF1A Q16665 1/20 0.47
FFAR4 Q5NUL3 1/20 0.47
CASP3 P42574 1/20 0.46
CASP6 P55212 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4261688 1.00 ADRB2 (0.56) ADRB2ADRB3ADRB1CYP2D6ADRA1D
SCHEMBL4255083 0.93 ADRB2 (0.54) ADRB2ADRB3ADRB1CYP2D6CYP3A4
SCHEMBL4255084 0.89 ADRB2 (0.57) ADRB2ADRB3ADRB1CYP2D6ADRA1D
SCHEMBL4261367 0.87 ADRB2 (0.53) ADRB2ADRB3ADRB1CYP2D6ADRA1D
SCHEMBL4389552 0.86 ADRB2 (0.54) ADRB2ADRB3ADRB1CYP2D6ADRA1D
SCHEMBL4389556 0.86 ADRB2 (0.54) ADRB2ADRB3ADRB1CYP2D6ADRA1D
SCHEMBL10662416 0.85 ADRB2 (0.52) ADRB2ADRB3ADRB1CYP2D6ADRA1D
SCHEMBL10662496 0.85 ADRB2 (0.52) ADRB2ADRB3ADRB1CYP2D6ADRA1D
SCHEMBL4255273 0.85 ADRB2 (0.72) ADRB2ADRB3ADRB1CASP3CASP6
SCHEMBL4257427 0.85 ADRB2 (0.72) ADRB2ADRB3ADRB1CASP3CASP6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1624868-B9 \"(2-HYDROXY-2-(4-HYDROXY-3-HYDOXYMETHYLPHENYL)-ETHYLAMINO)- PROPYL]PHENYL DERIVATIVES AS BETA2 AGONISTS PFIZER LTD (GB) 2009-08-12 EP claimed
EP-1624868-B1 \"(2-HYDROXY-2-(4-HYDROXY-3-HYDOXYMETHYLPHENYL)-ETHYLAMINO)- PROPYL]PHENYL DERIVATIVES AS BETA2 AGONISTS PFIZER LTD (GB) 2008-11-12 EP claimed