SCHEMBL4263449

SCHEMBL4263449

CC(C=O)=CC1=C(Cl)c2ccccc2CC1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.49
MAPT P10636 3/20 0.46
GAA P10253 1/20 0.43
TSHR P16473 2/20 0.42
ALDH1A1 P00352 2/20 0.42
TDP1 Q9NUW8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CES1 P23141 1/20 0.38
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
PTAFR P25105 1/20 0.36
MAOB P27338 1/20 0.35
LMNA P02545 2/20 0.35
CYP3A4 P08684 2/20 0.35
SLC6A2 P23975 2/20 0.35
TP53 P04637 1/20 0.35
CYP1A2 P05177 1/20 0.35
ADRB2 P07550 1/20 0.35
RET P07949 1/20 0.35
CHRM2 P08172 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4263444 1.00 ESR1 (0.49) ESR1MAPTGAATSHRALDH1A1
SCHEMBL4271682 0.83 RAB9A (0.46) ESR1MAPTGAATDP1L3MBTL1
SCHEMBL4269301 0.83 RAB9A (0.46) ESR1MAPTGAATDP1L3MBTL1
SCHEMBL2063760 0.79 ESR1 (0.54) ESR1MAPTGAATDP1L3MBTL1
SCHEMBL29952458 0.79 ESR1 (0.54) ESR1MAPTGAATDP1L3MBTL1
SCHEMBL4412530 0.77 MAPT (0.43) ESR1MAPTGAAALDH1A1TDP1
SCHEMBL4412532 0.77 MAPT (0.43) ESR1MAPTGAAALDH1A1TDP1
SCHEMBL4410195 0.74 MAPT (0.41) ESR1MAPTGAAALDH1A1TDP1
SCHEMBL4410193 0.74 MAPT (0.41) ESR1MAPTGAAALDH1A1TDP1
SCHEMBL2063819 0.74 ESR1 (0.66) ESR1MAPTGAATDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009110002-A1 NOVEL EFFLUX PUMP INHIBITORS COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2009-09-11 WO disclosed