SCHEMBL4267036

SCHEMBL4267036

ClCCN(C=Cc1ccccc1)CCCl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.41
RELA Q04206 1/20 0.36
GRM5 P41594 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
ALDH1A1 P00352 2/20 0.35
LMNA P02545 2/20 0.35
MAPK1 P28482 2/20 0.35
NFE2L2 Q16236 1/20 0.35
CYP19A1 P11511 1/20 0.35
MAOA P21397 1/20 0.35
TRPA1 O75762 1/20 0.35
ALOX5 P09917 1/20 0.35
IDO1 P14902 2/20 0.35
PAM P19021 1/20 0.35
MAPT P10636 2/20 0.34
RECQL P46063 2/20 0.34
HDAC3 O15379 1/20 0.34
TNKS O95271 1/20 0.34
HDAC4 P56524 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10626718 0.79 NPC1 (0.42) MAOBRELAGRM5MEN1KMT2A
SCHEMBL4267199 0.76 BCHE (0.42) MAOBRELAGRM5MEN1KMT2A
SCHEMBL4831765 0.75 EGFR (0.43) RELALMNAMAPTHDAC3SMN1; SMN2
Boric Acid SCHEMBL28492772 0.75 CA1 (0.44) MAOBRELAKMT2AALDH1A1LMNA
SCHEMBL11171879 0.74 NPC1 (0.48) MAOBRELAGRM5TRPA1NPC1
SCHEMBL136178 0.74 NPC1 (0.48) MAOBRELAGRM5TRPA1NPC1
SCHEMBL10628700 0.73 EGFR (0.45) LMNAMAPTHDAC3SMN1; SMN2NPC1
SCHEMBL303152 0.73 EGFR (0.45) LMNAMAPTHDAC3SMN1; SMN2NPC1
SCHEMBL10623988 0.73 EGFR (0.45) LMNAMAPTHDAC3SMN1; SMN2NPC1
SCHEMBL10628492 0.73 EGFR (0.45) LMNAMAPTHDAC3SMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9133195-B2 Quaternary ammonium salt compounds of spirocyclopiperazines, preparation methods and uses thereof PEKING UNIVERSITY (CN) 2015-09-15 US disclosed
US-20090325929-A1 QUATERNARY AMMONIUM SALT COMPOUNDS OF SPIROCYCLOPIPERAZINES, PREPARATION METHODS AND USES THEREOF PEKING UNIVERSITY (CN) 2009-12-31 US disclosed
EP-2036909-A1 QUATERNARY AMMONIUM SALT COMPOUNDS OF SPIROCYCLOPIPERAZINES, PREPARATION METHODS AND USES THEREOF Peking University (CN) 2009-03-18 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090325929-A1 QUATERNARY AMMONIUM SALT COMPOUNDS OF SPIROCYCLOPIPERAZINES, PREPARATION METHODS AND USES THEREOF CHRM4, CHRM1, CHRNA4 MAOB 1221/4885RELA 1710/4885GRM5 87/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.