SCHEMBL4276252

SCHEMBL4276252

O=C(Nc1ncc(CCc2ccccc2)s1)c1ccc2c(c1)CCNC2

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.48
FDPS P14324 1/20 0.45
TP53 P04637 2/20 0.44
OGA O60502 1/20 0.44
GAA P10253 1/20 0.44
WNT1 P04628 2/20 0.43
GSK3B P49841 2/20 0.43
DYRK1A Q13627 2/20 0.43
CLK2 P49760 1/20 0.43
CLK3 P49761 1/20 0.43
CYP3A4 P08684 1/20 0.42
ROCK2 O75116 1/20 0.42
MAPT P10636 3/20 0.42
F2 P00734 1/20 0.42
PLG P00747 1/20 0.42
PLAU P00749 1/20 0.42
PLAT P00750 1/20 0.42
KLKB1 P03952 1/20 0.42
PRSS1 P07477 1/20 0.42
KMT2A Q03164 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4289740 0.99 POLB (0.47) POLBFDPSTP53OGAGAA
SCHEMBL4283271 0.91 POLB (0.56) POLBTP53GAAMAPTKMT2A
SCHEMBL4563945 0.84 POLB (0.48) POLBTP53OGAGAAWNT1
SCHEMBL3738441 0.83 NPC1 (0.62) POLBKMT2AMEN1NPC1ALDH1A1
SCHEMBL4288598 0.83 KMT2A (0.61) POLBTP53GAACYP3A4MAPT
Hydrochloric Acid SCHEMBL3731968 0.83 NPC1 (0.61) POLBKMT2AMEN1NPC1ALDH1A1
Hydrochloric Acid SCHEMBL4279918 0.83 KMT2A (0.60) POLBTP53GAACYP3A4MAPT
SCHEMBL4285057 0.82 MAPT (0.60) POLBGAACYP3A4MAPTKMT2A
SCHEMBL4284053 0.82 GAA (0.57) GAACYP3A4MAPTKMT2ACYP1A2
Hydrochloric Acid SCHEMBL4279689 0.81 MAPT (0.59) POLBGAACYP3A4MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009150196-A1 N-THIAZOLYL-1, 2, 3, 4-TETRAHYDRO-6-ISOQUINOLINECARBOXAMIDE DERIVATIVES AS INHIBITORS OF STEAROYL COENZYME A DESATURASE SMITHKLINE BEECHAM CORPORATION (US) 2009-12-17 WO claimed
WO-2009150196-A1 N-THIAZOLYL-1, 2, 3, 4-TETRAHYDRO-6-ISOQUINOLINECARBOXAMIDE DERIVATIVES AS INHIBITORS OF STEAROYL COENZYME A DESATURASE SMITHKLINE BEECHAM CORPORATION (US) 2009-12-17 WO disclosed