SCHEMBL4285057

SCHEMBL4285057

O=C(Nc1ncc(Cc2ccccc2Cl)s1)c1ccc2c(c1)CCNC2

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.60
MEN1 O00255 5/20 0.58
KMT2A Q03164 5/20 0.58
LMNA P02545 3/20 0.58
TDP1 Q9NUW8 1/20 0.58
L3MBTL1 Q9Y468 1/20 0.58
ABL1 P00519 3/20 0.55
POLB P06746 2/20 0.53
ALDH1A1 P00352 2/20 0.51
CFTR P13569 1/20 0.51
KDM4E B2RXH2 1/20 0.51
SMN1; SMN2 Q16637 4/20 0.50
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
GAA P10253 2/20 0.49
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C19 P33261 1/20 0.48
HTT P42858 1/20 0.48
PKM P14618 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4279689 0.99 MAPT (0.59) MAPTMEN1KMT2ALMNATDP1
SCHEMBL4284162 0.90 MAPT (0.61) MAPTMEN1KMT2ALMNATDP1
Hydrochloric Acid SCHEMBL4279963 0.89 MAPT (0.60) MAPTMEN1KMT2ALMNATDP1
SCHEMBL4281317 0.88 LMNA (0.51) MAPTMEN1KMT2ALMNATDP1
SCHEMBL4283271 0.87 POLB (0.56) MAPTMEN1KMT2ALMNAL3MBTL1
Hydrochloric Acid SCHEMBL4288617 0.87 LMNA (0.50) MAPTMEN1KMT2ALMNATDP1
SCHEMBL4281323 0.85 SCD (0.56) MAPTMEN1KMT2ALMNASMN1; SMN2
SCHEMBL4284053 0.85 GAA (0.57) MAPTMEN1KMT2ALMNAL3MBTL1
SCHEMBL4288598 0.85 KMT2A (0.61) MAPTMEN1KMT2ALMNAABL1
Hydrochloric Acid SCHEMBL4289761 0.85 SCD (0.56) MAPTMEN1KMT2ALMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009150196-A1 N-THIAZOLYL-1, 2, 3, 4-TETRAHYDRO-6-ISOQUINOLINECARBOXAMIDE DERIVATIVES AS INHIBITORS OF STEAROYL COENZYME A DESATURASE SMITHKLINE BEECHAM CORPORATION (US) 2009-12-17 WO claimed
WO-2009150196-A1 N-THIAZOLYL-1, 2, 3, 4-TETRAHYDRO-6-ISOQUINOLINECARBOXAMIDE DERIVATIVES AS INHIBITORS OF STEAROYL COENZYME A DESATURASE SMITHKLINE BEECHAM CORPORATION (US) 2009-12-17 WO disclosed