SCHEMBL4276284

SCHEMBL4276284

CC(C)(C)N1CCC2(CC1)CC(O[Si](C)(C)C(C)(C)C)c1cc(-c3noc(=O)[nH]3)ccc1O2

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
RARB P10826 2/20 0.33
RARG P13631 1/20 0.33
PLA2G2A P14555 5/20 0.33
ALDH1A1 P00352 1/20 0.32
RBP4 P02753 1/20 0.32
RARA P10276 1/20 0.31
XDH P47989 1/20 0.31
IP6K1 Q92551 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL733219 0.89 RBP4 (0.35) RARBRARGPLA2G2AALDH1A1RBP4
SCHEMBL309170 0.87 IDO1 (0.41) RBP4
SCHEMBL1815579 0.87 IDO1 (0.41) RBP4
SCHEMBL310131 0.73 IDO1 (0.43) RBP4
SCHEMBL1812127 0.73 IDO1 (0.43) RBP4
SCHEMBL731730 0.71 HDAC3 (0.39) RARBRARGPLA2G2ARBP4RARA
SCHEMBL732818 0.66 IDO1 (0.43)
SCHEMBL309247 0.65 KMT2A (0.49) ALDH1A1
SCHEMBL743373 0.64 IDO1 (0.43)
SCHEMBL732811 0.64 IDO1 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2120569-A2 SPIROCHROMANON DERIVATIVES Merck & Co., Inc. (US) 2009-11-25 EP disclosed
WO-2008088692-A2 SPIROCHROMANON DERIVATIVES MERCK & CO., INC. (US) 2008-07-24 WO disclosed