SCHEMBL4276308

SCHEMBL4276308

COc1cc(C(=O)[C@@H]2C(=O)c3cc(-c4cncc(C(=O)O)c4)ccc3OC23CCNCC3)cc(OC)c1-c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACB O00763 1/20 0.43
ACACA Q13085 1/20 0.43
OPRD1 P41143 2/20 0.34
CYP1A1 P04798 1/20 0.33
CYP1B1 Q16678 1/20 0.33
ITGA4 P13612 1/20 0.33
ITGB7 P26010 1/20 0.33
BRD4 O60885 1/20 0.33
NR1H4 Q96RI1 2/20 0.32
OPRK1 P41145 1/20 0.32
KCNH2 Q12809 1/20 0.32
PDE4A P27815 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE4C Q08493 1/20 0.31
PDE4D Q08499 1/20 0.31
MKNK1 Q9BUB5 2/20 0.31
MKNK2 Q9HBH9 2/20 0.31
RARA P10276 1/20 0.30
RARB P10826 1/20 0.30
RARG P13631 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4412902 0.86 ACACB (0.41) ACACBACACABRD4MKNK1MKNK2
SCHEMBL3864125 0.84 ACACB (0.54) ACACBACACACYP1A1CYP1B1
SCHEMBL3793047 0.84 ACACB (0.51) ACACBACACACYP1A1CYP1B1
SCHEMBL1444711 0.84 ACACB (0.51) ACACBACACACYP1A1CYP1B1
SCHEMBL4266728 0.83 OPRD1 (0.32) ACACBOPRD1ITGA4ITGB7OPRK1
SCHEMBL4267712 0.83 OPRD1 (0.32) ACACBOPRD1ITGA4ITGB7OPRK1
SCHEMBL4416789 0.83 ACACB (0.38) ACACBACACAMKNK1MKNK2SSTR5
SCHEMBL14128719 0.83 ACACB (0.66) ACACBACACACYP1A1CYP1B1
SCHEMBL2571790 0.83 ACACB (0.66) ACACBACACACYP1A1CYP1B1
SCHEMBL4266808 0.83 OPRD1 (0.32) ACACBOPRD1ITGA4ITGB7OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2120569-A2 SPIROCHROMANON DERIVATIVES Merck & Co., Inc. (US) 2009-11-25 EP claimed
WO-2008088692-A2 SPIROCHROMANON DERIVATIVES MERCK & CO., INC. (US) 2008-07-24 WO claimed