Medroxyprogesterone Acetate

Medroxyprogesterone Acetate

SCHEMBL4277

CC(=O)O.CC(=O)O[C@]1(C(C)=O)CC[C@H]2[C@@H]3C[C@H](C)C4=CC(=O)CC[C@]4(C)[C@H]3CC[C@@]21C

nearest known ligand 0.96

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

PGR

The experimentally established mechanism targets of Medroxyprogesterone Acetate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR known ✓ P06401 4/20 0.96
NR3C1 P04150 5/20 0.96
LMNA P02545 4/20 0.96
CYP3A4 P08684 4/20 0.96
AR P10275 4/20 0.96
SMN1; SMN2 Q16637 4/20 0.96
NPSR1 Q6W5P4 3/20 0.96
ABCB11 O95342 2/20 0.96
ALDH1A1 P00352 2/20 0.96
CHRM2 P08172 2/20 0.96
CHRM1 P11229 2/20 0.96
USP2 O75604 2/20 0.96
SHBG P04278 2/20 0.96
ABCC4 O15439 1/20 0.96
ESR1 P03372 1/20 0.96
NR3C2 P08235 1/20 0.96
HRH2 P25021 1/20 0.96
AKR1C3 P42330 1/20 0.96
AKR1C2 P52895 1/20 0.96
AKR1C1 Q04828 1/20 0.96

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Medroxyprogesterone Acetate SCHEMBL4556265 1.00 NR3C1 (0.96) NR3C1LMNACYP3A4PGRAR
Medroxyprogesterone Acetate SCHEMBL5493761 1.00 NR3C1 (0.96) NR3C1LMNACYP3A4PGRAR
Medroxyprogesterone Acetate SCHEMBL8987454 1.00 NR3C1 (0.96) NR3C1LMNACYP3A4PGRAR
Medroxyprogesterone Acetate SCHEMBL10080145 0.98 NR3C1 (1.00) NR3C1LMNACYP3A4PGRAR
Medroxyprogesterone Acetate SCHEMBL3892232 0.98 NR3C1 (1.00) NR3C1LMNACYP3A4PGRAR
Medroxyprogesterone Acetate SCHEMBL6835475 0.98 NR3C1 (1.00) NR3C1LMNACYP3A4PGRAR
Medroxyprogesterone Acetate SCHEMBL4276 0.98 NR3C1 (1.00) NR3C1LMNACYP3A4PGRAR
Medroxyprogesterone Acetate SCHEMBL6563018 0.98 NR3C1 (1.00) NR3C1LMNACYP3A4PGRAR
Medroxyprogesterone Acetate SCHEMBL22761990 0.98 NR3C1 (1.00) NR3C1LMNACYP3A4PGRAR
Medroxyprogesterone Acetate SCHEMBL13941346 0.98 NR3C1 (1.00) NR3C1LMNACYP3A4PGRAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 34198 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116209439-B Cereblon protein modulators Saint Jude Children's Research Hospital Ltd. (US) 2026-05-26 CN claimed
CN-122084582-A Auxiliary kit for detecting content of calcium ions in cells 2026-05-26 CN claimed
WO-2026097604-A1 COMPOSITION AND DRUG-DEVICE COMBINATION PRODUCT FOR LOCAL TUMOR ADMINISTRATION, AND USE 诺曼德美国有限责任公司 2026-05-15 WO claimed
EP-3773730-B1 DRUG DELIVERY FORMULATIONS UNIV CALIFORNIA (US) 2026-05-13 EP claimed
US-20260109699-A1 AZOLE DERIVATIVES AS SHP2 INHIBITORS IRBM S.P.A. (IT) 2026-04-23 US claimed
US-20260097039-A1 METHODS FOR TREATING A FATTY LIVER DISEASE MADRIGAL PHARMACEUTICALS INC (US) 2026-04-09 US claimed
US-20260091119-A1 ISOLATED TARGETED DELIVERY SYSTEM FOR THE TREATMENT OF GLIOMA CELLIS AG (CH) 2026-04-02 US claimed
EP-4711364-A1 FUSED PYRROLE RING OR FUSED PYRIDINE RING COMPOUND Pharmaengine, Inc. (TW) 2026-03-18 EP claimed
US-12577255-B2 MDM2-based modulators of proteolysis and associated methods of use ARVINAS OPERATIONS, INC. (US) 2026-03-17 US claimed
EP-4704832-A2 BIFUNCTIONAL SMALL MOLECULES TO TARGET THE SELECTIVE DEGRADATION OF CIRCULATING PROTEINS Biohaven Therapeutics Ltd. (VG) 2026-03-11 EP claimed
EP-0163489-A1 Treatment of female hair loss Mortimer, Christopher Harry, Dr. (GB) 1985-12-04 EP claimed
EP-0136781-A2 Treatment of endometriosis AMERICAN HOME PRODUCTS CORPORATION (US) 1985-04-10 EP claimed
EP-0123528-A1 Pharmaceutical composition for the treatment of hair loss Mortimer, Christopher Harry, Dr. (GB) 1984-10-31 EP claimed
WO-1984004038-A1 PHARMACEUTICAL COMPOSITION FOR THE TREATMENT OF HAIR LOSS MORTIMER CHRISTOPHER HARRY (GB) 1984-10-25 WO claimed
EP-0114003-A1 Antiandrogen and antibiotic treatment of acne and pharmaceutical preparations therefor Mortimer, Christopher Harry, Dr. (GB) 1984-07-25 EP claimed
US-4310510-A Self administrable anti-fertility composition SHERMAN KENNETH N 1982-01-12 US claimed
US-4252787-A CONTRACEPTIVES, PROGESTATIONAL ACTIVITY, STEROIDS CAMBRIDGE RESEARCH AND DEVELOPMENT GROUP (US) 1981-02-24 US claimed
US-4038389-A VEHICLE FOR PARENTERAL ADMINISTRATION THE UPJOHN COMPANY (US) 1977-07-26 US claimed
US-3942641-A Dispensing packages containing novel cyclic progestogen-interrupted estrogen oral contraceptive regimens SYNTEX CORPORATION (PM) 1976-03-09 US claimed
US-3932635-A Novel cyclic progestogen-interrupted estrogen oral contraceptive regimens SYNTEX CORPORATION (PM) 1976-01-13 US claimed