SCHEMBL4277338

SCHEMBL4277338

CNc1ncc2c(c1C(C)(C)C)NC(=O)N(c1ccc(F)c(NC(=O)Nc3cc(C(C)(C)C)no3)c1)C2

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 3/20 0.47
KDR P35968 3/20 0.47
RAF1 P04049 3/20 0.47
KRAS P01116 2/20 0.47
MAP2K2 P36507 2/20 0.47
MAP2K1 Q02750 2/20 0.47
MAPK14 Q16539 8/20 0.41
MAPK13 O15264 2/20 0.39
ALDH1A1 P00352 1/20 0.39
NTRK1 P04629 2/20 0.38
NTRK3 Q16288 1/20 0.38
NTRK2 Q16620 1/20 0.38
CNR2 P34972 3/20 0.38
CSF1R P07333 1/20 0.37
RET P07949 1/20 0.36
EPHB2 P29323 1/20 0.36
CYP2C8 P10632 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
FLT3 P36888 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4271182 0.81 BRAF (0.43) BRAFKDRRAF1KRASMAP2K2
SCHEMBL4562970 0.80 BRAF (0.42) BRAFKDRRAF1KRASMAP2K2
SCHEMBL1521767 0.80 BRAF (0.53) BRAFKDRRAF1KRASMAP2K2
SCHEMBL1521806 0.79 BRAF (0.46) BRAFKDRRAF1KRASMAP2K2
SCHEMBL4276058 0.79 BRAF (0.45) BRAFKDRRAF1KRASMAP2K2
SCHEMBL1521899 0.79 BRAF (0.52) BRAFKDRRAF1KRASMAP2K2
SCHEMBL4273927 0.79 BRAF (0.52) BRAFKDRRAF1KRASMAP2K2
SCHEMBL1522009 0.78 BRAF (0.56) BRAFKDRRAF1KRASMAP2K2
SCHEMBL1521795 0.78 BRAF (0.47) BRAFKDRRAF1KRASMAP2K2
SCHEMBL1521556 0.77 BRAF (0.52) BRAFKDRRAF1KRASMAP2K2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2063896-A2 KINASE INHIBITORS USEFUL FOR THE TREATMENT OF PROLIFERATIVE DISEASES Deciphera Pharmaceuticals, LLC. (US) 2009-06-03 EP disclosed
WO-2008033999-A2 KINASE INHIBITORS USEFUL FOR THE TREATMENT OF PROLIFERATIVE DISEASES DECIPHERA PHARMACEUTICALS, LLC (US) 2008-03-20 WO disclosed