SCHEMBL4277652

SCHEMBL4277652

Cc1ccccc1S(=O)(=O)Nc1ccc2ccccc2c1C(=O)O

nearest known ligand 0.69

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 3/20 0.69
METAP1 P53582 1/20 0.69
SLC40A1 Q9NP59 1/20 0.48
TSHR P16473 1/20 0.47
MEN1 O00255 4/20 0.47
KMT2A Q03164 4/20 0.47
HCRTR1 O43613 1/20 0.46
BRD4 O60885 1/20 0.46
MCL1 Q07820 1/20 0.45
ALDH1A1 P00352 1/20 0.45
HPGD P15428 1/20 0.45
HSD17B10 Q99714 1/20 0.45
GAA P10253 1/20 0.44
G6PD P11413 1/20 0.44
MAP1LC3B Q9GZQ8 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3985999 0.88 METAP2 (0.74) METAP2METAP1TSHRMEN1KMT2A
SCHEMBL3982685 0.86 METAP2 (0.67) METAP2METAP1MEN1KMT2AMCL1
SCHEMBL3985482 0.84 METAP2 (0.69) METAP2METAP1TSHRMEN1KMT2A
SCHEMBL3979302 0.84 METAP2 (0.69) METAP2METAP1TSHRMEN1KMT2A
SCHEMBL3986500 0.82 METAP2 (1.00) METAP2METAP1MEN1KMT2AMCL1
SCHEMBL3986006 0.82 METAP2 (0.62) METAP2METAP1SLC40A1TSHRMEN1
SCHEMBL3984291 0.82 METAP2 (0.82) METAP2METAP1TSHRALDH1A1
SCHEMBL3982643 0.81 METAP2 (0.60) METAP2METAP1TSHRMEN1KMT2A
SCHEMBL3982644 0.81 METAP2 (0.60) METAP2METAP1
SCHEMBL3982567 0.80 METAP2 (0.71) METAP2METAP1MEN1KMT2AMCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040068012-A1 Sulfonamides having antiangiogenic and anticancer activity ABBOTT LABORATORIES 2004-04-08 US claimed
US-7491718-B2 Sulfonamides having antiangiogenic and anticancer activity ABBOTT LABORATORIES (US) 2009-02-17 US disclosed
US-20040167128-A1 Sulfonamides having antiangiogenic and anticancer activity ABBVIE INC. 2004-08-26 US disclosed
US-20040157836-A1 Sulfonamides having antiangiogenic and anticancer activity ABBOTT LABORATORIES 2004-08-12 US disclosed
US-20040068012-A1 Sulfonamides having antiangiogenic and anticancer activity ABBOTT LABORATORIES 2004-04-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040167128-A1 Sulfonamides having antiangiogenic and anticancer activity METAP2, METAP1, DNPEP METAP2 1/4885METAP1 2/4885SLC40A1 3138/4885
US-20040068012-A1 Sulfonamides having antiangiogenic and anticancer activity METAP2, METAP1, DNPEP METAP2 1/4885METAP1 2/4885SLC40A1 3138/4885
US-20040157836-A1 Sulfonamides having antiangiogenic and anticancer activity METAP2, METAP1, DNPEP METAP2 1/4885METAP1 2/4885SLC40A1 3138/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.