SCHEMBL4278142

SCHEMBL4278142

CCOC(=O)[C@H](CCCC(F)(F)F)NC(=O)OC(C)(C)C

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.54
CYP2C9 P11712 1/20 0.54
CYP2C19 P33261 1/20 0.54
HTT P42858 1/20 0.54
CTSK P43235 9/20 0.49
SMN1; SMN2 Q16637 1/20 0.47
CTSS P25774 3/20 0.47
ALDH1A1 P00352 3/20 0.45
MAPT P10636 3/20 0.45
KDM4E B2RXH2 1/20 0.42
GAA P10253 1/20 0.42
PKM P14618 1/20 0.42
HPGD P15428 1/20 0.42
ALOX12 P18054 1/20 0.42
KMT2A Q03164 2/20 0.41
POLB P06746 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31390053 0.94 CYP1A2 (0.57) CYP1A2CYP2C9CYP2C19HTTCTSK
SCHEMBL30352865 0.89 CYP1A2 (0.53) CYP1A2CYP2C9CYP2C19HTTCTSK
SCHEMBL31341192 0.88 CTSK (0.48) CYP1A2CYP2C9CYP2C19HTTCTSK
SCHEMBL31075393 0.87 CYP1A2 (0.56) CYP1A2CYP2C9CYP2C19HTTCTSK
SCHEMBL24387324 0.87 CYP1A2 (0.56) CYP1A2CYP2C9CYP2C19HTTCTSK
SCHEMBL29399499 0.85 CYP1A2 (0.59) CYP1A2CYP2C9CYP2C19HTTCTSK
SCHEMBL18109724 0.84 CTSK (0.50) CTSKCTSSALDH1A1GAAKMT2A
SCHEMBL31036530 0.84 CTSK (0.50) CTSKCTSSALDH1A1GAAKMT2A
SCHEMBL18109722 0.84 CTSK (0.50) CTSKCTSSALDH1A1GAAKMT2A
SCHEMBL28766288 0.84 CTSK (0.55) CTSKCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1863812-A4 DIPEPTIDYL PEPTIDASE-IV INHIBITING COMPOUNDS, METHODS OF PREPARING THE SAME, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AS AN ACTIVE AGENT LG LIFE SCIENCES LTD (KR) 2009-06-24 EP disclosed
EP-1863812-A1 DIPEPTIDYL PEPTIDASE-IV INHIBITING COMPOUNDS, METHODS OF PREPARING THE SAME, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AS AN ACTIVE AGENT LG Life Sciences Ltd. (KR) 2007-12-12 EP disclosed
WO-2006104356-A1 DIPEPTIDYL PEPTIDASE-IV INHIBITING COMPOUNDS, METHODS OF PREPARING THE SAME, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AS AN ACTIVE AGENT LG LIFE SCIENCES, LTD. (KR) 2006-10-05 WO disclosed