Rogletimide

Rogletimide

SCHEMBL4281

CCC1(c2ccncc2)CCC(=O)NC1=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 19/20 1.00
CYP3A4 P08684 2/20 0.68
CYP17A1 P05093 1/20 0.68
CYP11A1 P05108 1/20 0.68
TBXAS1 P24557 1/20 0.68
PMP22 Q01453 1/20 0.68
PDE4D Q08499 1/20 0.68
PDE3A Q14432 1/20 0.68
NFKB1 P19838 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Rogletimide SCHEMBL9372682 1.00 CYP19A1 (1.00) CYP19A1CYP3A4CYP17A1CYP11A1TBXAS1
Rogletimide SCHEMBL28110686 0.97 CYP19A1 (0.94) CYP19A1CYP3A4CYP17A1CYP11A1TBXAS1
SCHEMBL3296751 0.85 CYP19A1 (1.00) CYP19A1
Glutethimide SCHEMBL113708 0.84 CYP19A1 (0.72) CYP19A1CYP3A4CYP17A1CYP11A1TBXAS1
Glutethimide SCHEMBL21119240 0.84 CYP19A1 (0.72) CYP19A1CYP3A4CYP17A1CYP11A1TBXAS1
Glutethimide SCHEMBL113709 0.84 CYP19A1 (0.72) CYP19A1CYP3A4CYP17A1CYP11A1TBXAS1
SCHEMBL9531145 0.83 CYP19A1 (1.00) CYP19A1
SCHEMBL16509358 0.83 CYP19A1 (0.75) CYP19A1CYP3A4CYP17A1CYP11A1TBXAS1
Aminoglutethimide SCHEMBL116988 0.81 CYP19A1 (1.00) CYP19A1CYP3A4CYP17A1CYP11A1TBXAS1
Aminoglutethimide SCHEMBL1230613 0.81 CYP19A1 (1.00) CYP19A1CYP3A4CYP17A1CYP11A1TBXAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 11417 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260116861-A1 ISOXAZOLE HYDROXAMIC ACIDS AS HISTONE DEACETYLASE 6 INHIBITORS THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-04-30 US claimed
US-12522572-B2 Isoxazole hydroxamic acids as histone deacetylase 6 inhibitors THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-01-13 US claimed
EP-4524131-A1 SMALL MOLECULES FOR TREATING CANCER, INHABITING CHEMOKINE ACTIVITY AND/OR INDUCING CELL DEATH AlonBio Ltd. (IL) 2025-03-19 EP claimed
US-12202803-B2 Small molecules for treating cancer, inhibiting chemokine activity and/or inducing cell death ALONBIO LTD. (IL) 2025-01-21 US claimed
US-20240343697-A1 ISOXAZOLE HYDROXAMIC ACIDS AS HISTONE DEACETYLASE 6 INHIBITORS THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2024-10-17 US claimed
US-12109219-B2 Cannabinoid receptor modulators ARENA PHARMACEUTICALS, INC. (US) 2024-10-08 US claimed
WO-2024026505-A2 DISRUPTION OF TELOCYTE ACTIVITY PATEL AMIT (US) 2024-02-01 WO claimed
US-20240002347-A1 SMALL MOLECULES FOR TREATING CANCER, INHIBITING CHEMOKINE ACTIVITY AND/OR INDUCING CELL DEATH ALONBIO LTD. (IL) 2024-01-04 US claimed
US-20220401541-A1 INTRATUMORAL ADMINISTRATION OF IMMUNE CELLULAR THERAPEUTICS FIBROBIOLOGICS, INC. 2022-12-22 US claimed
EP-3441089-B1 TREATMENT METHODS USING ADENOVIRUS VASCULAR BIOGENICS LTD (IL) 2022-12-14 EP claimed
EP-1019034-A2 ANTIOXIDANT ENHANCEMENT OF THERAPY FOR HYPERPROLIFERATIVE CONDITIONS Atherogenics, Inc. (US) 2000-07-19 EP claimed
US-6020327-A Control of hair growth THE CENTRAL SHEFFIELD UNIVERSITY HOSPITALS NHS TRUST (GB) 2000-02-01 US claimed
WO-1999001118-A9 ANTIOXIDANT ENHANCEMENT OF THERAPY FOR HYPERPROLIFERATIVE CONDITIONS ATHEROGENICS INC (US) 1999-05-20 WO claimed
WO-1999001118-A2 ANTIOXIDANT ENHANCEMENT OF THERAPY FOR HYPERPROLIFERATIVE CONDITIONS ATHEROGENICS, INC. (US) 1999-01-14 WO claimed
EP-0516278-A1 Use of anti-mullerian hormone for reversal of female sexual phenotype in poultry MERCK & CO. INC. (US) 1992-12-02 EP claimed
EP-0514015-A1 Control of sex differentiation in fish MERCK & CO. INC. (US) 1992-11-19 EP claimed
US-5162337-A Administering Steroid Biosynthesis Inhibitors MERCK & CO., INC. (US) 1992-11-10 US claimed
WO-1992018132-A1 PHARMACEUTICAL COMBINATION FOR THE TREATMENT OF BENIGN PROSTATIC HYPERPLASIA COMTAINING A 5 ALPHA-REDUCTASE INHIBITOR MERCK & CO., INC. (US) 1992-10-29 WO claimed
EP-0479570-A2 Animal growth promotion with aromatase inhibitors MERCK & CO. INC. (US) 1992-04-08 EP claimed
EP-0433084-A2 Use of aromatese inhibitors for the reversal of female sexual phenotype in poultry MERCK & CO. INC. (US) 1991-06-19 EP claimed