SCHEMBL4283013

SCHEMBL4283013

COC(=O)c1c(C)cc(C=O)cc1C

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.52
ACHE P22303 1/20 0.52
ALDH1A1 P00352 7/20 0.50
HPGD P15428 3/20 0.49
SRC P12931 1/20 0.46
PTGES O14684 1/20 0.46
PTPN1 P18031 1/20 0.46
POLB P06746 2/20 0.44
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
CA14 Q9ULX7 1/20 0.41
RAB9A P51151 1/20 0.41
GLO1 Q04760 1/20 0.40
USP2 O75604 1/20 0.39
ATM Q13315 1/20 0.39
TRIM24 O15164 1/20 0.39
ALDH5A1 P51649 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22890563 0.88 CYP3A4 (0.45) CYP3A4ACHEALDH1A1HPGDSRC
SCHEMBL1515913 0.82 ALDH1A1 (0.50) CYP3A4ACHEALDH1A1HPGDPTGES
SCHEMBL9100361 0.80 ALDH1A1 (0.50) CYP3A4ACHEALDH1A1HPGDPOLB
SCHEMBL22032247 0.79 SRC (0.42) CYP3A4ACHEALDH1A1HPGDSRC
SCHEMBL1036031 0.79 CYP3A4 (0.59) CYP3A4ACHEALDH1A1HPGDPOLB
SCHEMBL879308 0.78 ALDH1A1 (0.48) CYP3A4ACHEALDH1A1HPGDPOLB
SCHEMBL14893350 0.78 ALDH1A1 (0.48) CYP3A4ACHEALDH1A1HPGDPTGES
SCHEMBL3308517 0.78 ALDH1A1 (0.44) CYP3A4ACHEALDH1A1HPGDSRC
SCHEMBL29017440 0.77 SRC (0.46) CYP3A4ALDH1A1HPGDSRCUSP2
SCHEMBL70139 0.77 CYP3A4 (0.57) CYP3A4ACHEALDH1A1HPGDPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009149795-A2 HETEROCYCLIC CYCLOPROPYL-SUBSTITUTED FXR BINDING COMPOUNDS PHENEX PHARMACEUTICALS AG (DE) 2009-12-17 WO disclosed
EP-2128158-A1 Heterocyclic cyclopropyl-substituted FXR binding compounds Phenex Pharmaceuticals AG (DE) 2009-12-02 EP disclosed