SCHEMBL4286559

SCHEMBL4286559

N#Cc1ccc2c(c1)CCN2C(=O)CCC(=O)O

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.62
CYP2C9 P11712 2/20 0.57
S1PR1 P21453 3/20 0.53
TSHR P16473 3/20 0.53
KMT2A Q03164 3/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
HPGD P15428 2/20 0.53
PTPN11 Q06124 3/20 0.52
S1PR4 O95977 1/20 0.51
S1PR5 Q9H228 1/20 0.51
MEN1 O00255 1/20 0.50
POLB P06746 4/20 0.49
GAA P10253 2/20 0.49
TDP1 Q9NUW8 2/20 0.49
ALDH1A1 P00352 2/20 0.49
HSD17B10 Q99714 1/20 0.49
CYP2C19 P33261 1/20 0.49
KDM4E B2RXH2 1/20 0.49
PTPN7 P35236 1/20 0.49
TP53 P04637 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3128299 0.86 TP53 (0.49) NOTUMCYP2C9S1PR1TSHRKMT2A
SCHEMBL3456314 0.83 TP53 (0.51) NOTUMTSHRKMT2ASMN1; SMN2HPGD
SCHEMBL4284878 0.82 NOTUM (0.49) NOTUMCYP2C9S1PR1TSHRKMT2A
SCHEMBL7814158 0.81 NOTUM (0.65) NOTUMCYP2C9TSHRKMT2ASMN1; SMN2
SCHEMBL20908660 0.81 NOTUM (0.65) NOTUMCYP2C9S1PR1TSHRKMT2A
SCHEMBL3457235 0.79 NOTUM (0.65) NOTUMKMT2ASMN1; SMN2HPGDMEN1
SCHEMBL21425395 0.79 CYP11B1 (0.48) NOTUMTDP1TP53MAPT
SCHEMBL20941553 0.77 TP53 (0.51) KMT2AMEN1POLBALDH1A1HSD17B10
SCHEMBL2278917 0.77 NOTUM (1.00) NOTUMTSHRKMT2ASMN1; SMN2MEN1
SCHEMBL31650229 0.77 NOTUM (1.00) NOTUMTSHRKMT2ASMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009151621-A1 SUBSTITUTED (1, 2, 4-0XADIAZ0L-3-YL) INDOLIN-1-YL CARBOXYLIC ACID DERIVATIVES USEFUL AS S1P1 AGONISTS ARENA PHARMACEUTICALS, INC. (US) 2009-12-17 WO disclosed