SCHEMBL4284878

SCHEMBL4284878

CC(C)(C)OC(=O)CCC(=O)N1CCc2cc(C#N)ccc21

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 6/20 0.49
TP53 P04637 1/20 0.46
GPR119 Q8TDV5 1/20 0.46
TSHR P16473 2/20 0.45
USP2 O75604 2/20 0.45
PKM P14618 1/20 0.45
ALDH1A1 P00352 1/20 0.44
S1PR1 P21453 3/20 0.44
DRD2 P14416 1/20 0.43
S1PR4 O95977 1/20 0.42
S1PR5 Q9H228 1/20 0.42
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
MEN1 O00255 1/20 0.40
MAPT P10636 1/20 0.40
KMT2A Q03164 1/20 0.40
CYP2C9 P11712 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13656966 0.83 GPR119 (0.47) NOTUMTP53GPR119DRD2CYP11B1
SCHEMBL4286559 0.82 NOTUM (0.62) NOTUMTP53TSHRALDH1A1S1PR1
SCHEMBL3128299 0.79 TP53 (0.49) NOTUMTP53TSHRUSP2ALDH1A1
SCHEMBL4279462 0.78 NOTUM (0.46) NOTUMTP53GPR119TSHRUSP2
SCHEMBL3456314 0.76 TP53 (0.51) NOTUMTP53TSHRUSP2ALDH1A1
SCHEMBL773073 0.76 DRD2 (0.64) ALDH1A1S1PR1DRD2MEN1MAPT
SCHEMBL3457235 0.75 NOTUM (0.65) NOTUMTP53ALDH1A1CYP11B1CYP11B2
SCHEMBL4284699 0.73 FNTA (0.41) GPR119DRD2
SCHEMBL21425395 0.72 CYP11B1 (0.48) NOTUMTP53CYP11B1CYP11B2MAPT
SCHEMBL3129984 0.71 CA12 (0.60) NOTUMTP53S1PR1S1PR4S1PR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009151621-A1 SUBSTITUTED (1, 2, 4-0XADIAZ0L-3-YL) INDOLIN-1-YL CARBOXYLIC ACID DERIVATIVES USEFUL AS S1P1 AGONISTS ARENA PHARMACEUTICALS, INC. (US) 2009-12-17 WO disclosed