SCHEMBL4288272

SCHEMBL4288272

N#CCCNC(=O)c1n[nH]cc1NC(=O)c1ccoc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTK2 Q05397 1/20 0.41
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
KCNK3 O14649 1/20 0.34
KCNK9 Q9NPC2 1/20 0.34
NOS3 P29474 1/20 0.34
NOS1 P29475 1/20 0.34
NOS2 P35228 1/20 0.34
TMIGD3 P0DMS9 1/20 0.33
ADORA1 P30542 1/20 0.33
RAB9A P51151 1/20 0.33
TBK1 Q9UHD2 1/20 0.32
CDK14 O94921 4/20 0.32
CCNY Q8ND76 4/20 0.32
PARP1 P09874 1/20 0.32
LRRK2 Q5S007 1/20 0.32
ITGAV P06756 2/20 0.31
MAPK14 Q16539 1/20 0.31
ADORA3 P0DMS8 1/20 0.31
EGFR P00533 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4283198 0.84 SMN1; SMN2 (0.40) HDAC3HDAC1RAB9ACDK14CCNY
SCHEMBL4294905 0.82 NPC1 (0.42) RAB9ACDK14CCNY
SCHEMBL4287676 0.80 KDM4E (0.42) HDAC1CDK14CCNYPARP1
SCHEMBL4288796 0.80 F10 (0.46) HDAC3HDAC1RAB9A
SCHEMBL4287274 0.80 ALDH1A1 (0.44) RAB9A
SCHEMBL4285709 0.79 GSK3B (0.48) HDAC1
SCHEMBL4288238 0.79 KMT2A (0.47) KCNK3KCNK9RAB9A
SCHEMBL4285079 0.79 CREBBP (0.42) HDAC1RAB9ACDK14CCNY
SCHEMBL4293174 0.79 MCHR1 (0.46) HDAC3
SCHEMBL4287235 0.78 MEN1 (0.52) RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090156582-A1 Pyrazole Compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-06-18 US disclosed
EP-1847531-A1 PYRAZOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2007-10-24 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090156582-A1 Pyrazole Compound GSK3B, GSK3A, GSKIP PTK2 1223/4885HDAC3 6/4885HDAC1 11/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.