SCHEMBL4288907

SCHEMBL4288907

Cc1nc(NC(=O)c2ccc3c(c2)CCNC3)sc1Cc1ccc(Cl)c(Cl)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 5/20 0.52
SMN1; SMN2 Q16637 5/20 0.52
ALDH1A1 P00352 5/20 0.52
LMNA P02545 3/20 0.52
KDM4E B2RXH2 3/20 0.52
HTT P42858 2/20 0.52
MAPT P10636 2/20 0.52
KMT2A Q03164 2/20 0.47
MEN1 O00255 1/20 0.47
NPSR1 Q6W5P4 2/20 0.44
RAB9A P51151 3/20 0.44
TDP1 Q9NUW8 1/20 0.44
CYP3A4 P08684 1/20 0.43
PTGER1 P34995 2/20 0.41
F2 P00734 1/20 0.41
PLG P00747 1/20 0.41
PLAU P00749 1/20 0.41
PLAT P00750 1/20 0.41
KLKB1 P03952 1/20 0.41
PRSS1 P07477 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4278242 0.99 HPGD (0.51) HPGDSMN1; SMN2ALDH1A1LMNAKDM4E
SCHEMBL4276192 0.91 HPGD (0.58) HPGDSMN1; SMN2ALDH1A1LMNAKDM4E
Hydrochloric Acid SCHEMBL4287252 0.90 HPGD (0.57) HPGDSMN1; SMN2ALDH1A1LMNAKDM4E
SCHEMBL4275912 0.89 SMN1; SMN2 (0.51) HPGDSMN1; SMN2ALDH1A1LMNAKDM4E
Hydrochloric Acid SCHEMBL4275235 0.88 SMN1; SMN2 (0.51) HPGDSMN1; SMN2ALDH1A1LMNAKDM4E
SCHEMBL4282184 0.87 HPGD (0.52) HPGDSMN1; SMN2ALDH1A1LMNAKDM4E
Hydrochloric Acid SCHEMBL4287316 0.86 HPGD (0.52) HPGDSMN1; SMN2ALDH1A1LMNAKDM4E
SCHEMBL13844946 0.86 SMN1; SMN2 (0.46) HPGDSMN1; SMN2ALDH1A1LMNAKDM4E
SCHEMBL4274873 0.86 SMN1; SMN2 (0.48) HPGDSMN1; SMN2ALDH1A1LMNAKDM4E
Hydrochloric Acid SCHEMBL4279972 0.85 SMN1; SMN2 (0.47) HPGDSMN1; SMN2ALDH1A1LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009150196-A1 N-THIAZOLYL-1, 2, 3, 4-TETRAHYDRO-6-ISOQUINOLINECARBOXAMIDE DERIVATIVES AS INHIBITORS OF STEAROYL COENZYME A DESATURASE SMITHKLINE BEECHAM CORPORATION (US) 2009-12-17 WO claimed