SCHEMBL4289698

SCHEMBL4289698

CN(C(=O)c1cnccn1)c1cn(C(c2ccccc2)(c2ccccc2)c2ccccc2)nc1C(=O)NC1CCCC1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
KMT2A Q03164 5/20 0.41
MAPT P10636 1/20 0.41
HTT P42858 2/20 0.39
GAA P10253 1/20 0.38
MEN1 O00255 3/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
SMYD3 Q9H7B4 1/20 0.37
GRM5 P41594 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CCNA2 P20248 1/20 0.36
CDK2 P24941 1/20 0.36
CCNA1 P78396 1/20 0.36
ACKR3 P25106 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4285857 0.84 TSHR (0.39) ALDH1A1GRM5CYP1A2CYP3A4CYP2D6
SCHEMBL4288801 0.83 HTT (0.39) ALDH1A1KMT2AHTTMEN1CYP1A2
SCHEMBL4286953 0.76 PDE10A (0.42) ALDH1A1MAPTCYP1A2CYP3A4CYP2C9
SCHEMBL4279856 0.70 RAB9A (0.43) ALDH1A1KMT2AMAPTHTTGAA
SCHEMBL4285067 0.68 TSHR (0.47) ALDH1A1KMT2AMAPTHTTMEN1
SCHEMBL12218526 0.66 GAA (0.64) ALDH1A1MAPTGAASMYD3GRM5
SCHEMBL20451349 0.66 GAA (0.64) ALDH1A1MAPTGAASMYD3GRM5
SCHEMBL28266316 0.65 SMYD3 (0.66) ALDH1A1KMT2AMAPTHTTGAA
SCHEMBL4289358 0.63 RAB9A (0.41) ALDH1A1KMT2AMAPTMEN1
SCHEMBL1535206 0.62 SMYD3 (0.74) ALDH1A1KMT2AMAPTHTTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090156582-A1 Pyrazole Compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-06-18 US disclosed
EP-1847531-A1 PYRAZOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2007-10-24 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090156582-A1 Pyrazole Compound GSK3B, GSK3A, GSKIP ALDH1A1 694/4885KMT2A 871/4885MAPT 868/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.