SCHEMBL4293047

SCHEMBL4293047

COc1cc(OC)c(OC)cc1C=CC#N

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 1/20 0.59
CYP3A4 P08684 1/20 0.59
NFE2L2 Q16236 2/20 0.52
CYP1A1 P04798 5/20 0.50
CYP1B1 Q16678 5/20 0.50
CYP1A2 P05177 4/20 0.50
KDM4E B2RXH2 2/20 0.50
ALDH1A1 P00352 2/20 0.50
TSHR P16473 2/20 0.50
FDPS P14324 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
ABCG2 Q9UNQ0 1/20 0.46
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
NOD2 Q9HC29 1/20 0.39
APP P05067 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15268735 0.85 FDPS (0.47) HMGCRCYP3A4NFE2L2CYP1A1CYP1B1
SCHEMBL15268738 0.85 FDPS (0.47) HMGCRCYP3A4NFE2L2CYP1A1CYP1B1
SCHEMBL7490539 0.83 PRKDC (0.55) HMGCRCYP3A4NFE2L2CYP1A1CYP1B1
SCHEMBL7490543 0.83 PRKDC (0.55) HMGCRCYP3A4NFE2L2CYP1A1CYP1B1
SCHEMBL3458624 0.82 HMGCR (0.41) HMGCRCYP3A4NFE2L2CYP1A1CYP1B1
SCHEMBL3458625 0.82 HMGCR (0.41) HMGCRCYP3A4NFE2L2CYP1A1CYP1B1
SCHEMBL333574 0.80 HMGCR (0.39) HMGCRCYP3A4NFE2L2CYP1A1CYP1B1
SCHEMBL333573 0.80 HMGCR (0.39) HMGCRCYP3A4NFE2L2CYP1A1CYP1B1
SCHEMBL2119648 0.80 HMGCR (0.59) HMGCRCYP3A4NFE2L2CYP1A1CYP1B1
SCHEMBL2119650 0.80 HMGCR (0.59) HMGCRCYP3A4NFE2L2CYP1A1CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1560837-B1 NOVEL AMPIPHILIC DERIVATIVES OF ALPHA-C-PHENYL N-TERT-BUTYL NITRONE TS PHARMA (FR) 2009-08-05 EP disclosed
EP-1560837-A2 NOVEL AMPIPHILIC DERIVATIVES OF ALPHA-C-PHENYL N-TERT-BUTYL NITRONE TS Pharma (FR) 2005-08-10 EP disclosed
WO-2004043982-A2 NOVEL AMPIPHILIC DERIVATIVES OF ALPHA-C-PHENYL N-TERT-BUTYL NITRONE TS PHARMA (FR) 2004-05-27 WO disclosed