SCHEMBL4293771

SCHEMBL4293771

O=C(CBr)c1ccc(OCc2ccccc2)c(NS(=O)(=O)CCc2ccccc2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.45
BCL2A1 Q16548 1/20 0.45
ACLY P53396 2/20 0.45
NPC1 O15118 1/20 0.44
HPGD P15428 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
PTGES2 Q9H7Z7 1/20 0.42
GLO1 Q04760 1/20 0.41
SMPD1 P17405 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
EGFR P00533 1/20 0.40
BRD4 O60885 3/20 0.40
PTPN1 P18031 1/20 0.40
PTGER1 P34995 1/20 0.39
PTGER4 P35408 1/20 0.39
PTGER3 P43115 1/20 0.39
PTGER2 P43116 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11880546 0.85 NPC1 (0.46) ACLYNPC1HPGDRAB9ASMN1; SMN2
SCHEMBL1221632 0.85 CYP19A1 (0.50) NPC1HPGDRAB9ASMN1; SMN2SMPD1
SCHEMBL6074414 0.84 SLC40A1 (0.51) MCL1BCL2A1ACLYNPC1HPGD
SCHEMBL7112677 0.83 AR (0.49) ACLYNPC1HPGDRAB9ASMN1; SMN2
SCHEMBL7107169 0.83 NPC1 (0.46) ACLYNPC1HPGDRAB9ASMN1; SMN2
SCHEMBL7111802 0.81 SMN1; SMN2 (0.47) ACLYNPC1HPGDRAB9ASMN1; SMN2
SCHEMBL7109250 0.81 NPC1 (0.48) NPC1HPGDRAB9ASMN1; SMN2SMPD1
SCHEMBL10451702 0.80 NPC1 (0.50) NPC1HPGDRAB9ASMN1; SMN2SMPD1
SCHEMBL8607319 0.80 CYP19A1 (0.56) NPC1HPGDRAB9ASMN1; SMN2HDAC1
SCHEMBL7109049 0.80 EGFR (0.45) ACLYNPC1HPGDRAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2035004-A1 PHENYL SUBSTITUTED PYRAZINOYLGUANIDINE SODIUM CHANNEL BLOCKERS POSSESSING BETA AGONIST ACTIVITY Parion Sciences, Inc. (US) 2009-03-18 EP disclosed
WO-2007146869-A1 PHENYL SUBSTITUTED PYRAZINOYLGUANIDINE SODIUM CHANNEL BLOCKERS POSSESSING BETA AGONIST ACTIVITY PARION SCIENCES, INC. (US) 2007-12-21 WO disclosed