SCHEMBL4300736

SCHEMBL4300736

CC(C(N)=O)N1CN([C@@H]2O[C@H](CO)C(O)C2O)c2nc(NCCc3ccc(CCC(=O)O)cc3)nc(N)c21

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 6/20 0.57
ADORA2B P29275 3/20 0.57
ADORA3 P0DMS8 2/20 0.52
KDM4E B2RXH2 3/20 0.44
ALOX15 P16050 2/20 0.44
HSD17B10 Q99714 2/20 0.44
KMT2A Q03164 2/20 0.44
ADORA1 P30542 1/20 0.44
TSHR P16473 1/20 0.44
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C19 P33261 1/20 0.44
PMP22 Q01453 1/20 0.43
ATM Q13315 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1081739 0.84 ADORA2A (0.57) ADORA2AADORA2BADORA3KDM4EALOX15
Hydrochloric Acid SCHEMBL6754870 0.84 ADORA2A (0.56) ADORA2AADORA2BADORA3KDM4EALOX15
Hydrochloric Acid SCHEMBL2031973 0.83 ADORA2A (0.55) ADORA2AADORA2BADORA3KDM4EALOX15
SCHEMBL13516554 0.82 ADORA2A (0.40) ADORA2AADORA2BADORA3ADORA1
SCHEMBL2295173 0.77 ADORA2A (0.48) ADORA2AADORA2BADORA3ADORA1
SCHEMBL724838 0.76 ADORA2A (0.47) ADORA2AADORA2BADORA3ADORA1
SCHEMBL726188 0.76 ADORA2A (0.46) ADORA2AADORA2BADORA3KDM4EALOX15
SCHEMBL846742 0.75 HSPA8 (0.46) ADORA2AADORA2BADORA3KDM4EALOX15
SCHEMBL940191 0.75 ADORA2A (0.46) ADORA2AADORA2BADORA3
SCHEMBL10588368 0.73 ADORA2A (1.00) ADORA2AADORA2BADORA3KDM4EALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-7082156-A None JP disclosed
US-20120197004-A1 NOVEL ANTI-MICROBIAL PEPTIDOMIMETIC COMPOUNDS AND METHODS TO CALCULATE ANTI-MICROBIAL ACTIVITY HICKS RICKEY P (US) 2012-08-02 US disclosed
US-8188033-B2 Anti-microbial peptidomimetic compounds and methods to calculate anti-microbial activity USA AS REPRESENTED BY THE SECRETARY OF THE ARMY ON BEHALF OF USAMRMC 2012-05-29 US disclosed
US-20090291898-A1 Novel anti-microbial peptidomimetic compounds and methods to calculate anti-microbial activity USA AS REPRESENTED BY THE SECRETARY OF THE ARMY ON BEHALF OF USAMRMC 2009-11-26 US disclosed
EP-2120983-A2 NOVEL ANTI-MICROBIAL PEPTIDOMIMETIC COMPOUNDS AND METHODS TO CALCULATE ANTI-MICROBIAL ACTIVITY The United States of America, as represented by The Secretary of the Army, on behalf of The Walter Reed Army Institute of Research (US) 2009-11-25 EP disclosed
WO-2008079314-A2 NOVEL ANTI-MICROBIAL PEPTIDOMIMETIC COMPOUNDS AND METHODS TO CALCULATE ANTI-MICROBIAL ACTIVITY THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY OF THE ARMY, ON BEHALF OF WALTER REED ARMY INSTITUTE OF RESEARCH (US) 2008-07-03 WO disclosed
JP-H0782156-A CANCER METASTASIS INHIBITOR NIPPON ZEON CO LTD 1995-03-28 JP disclosed