SCHEMBL4302963

SCHEMBL4302963

O=C(NCCc1ccc(F)cc1)c1cnc(C(=O)O)c(O)c1CO

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.46
RAB9A P51151 6/20 0.46
KMT2A Q03164 1/20 0.46
MAPT P10636 1/20 0.45
SMN1; SMN2 Q16637 3/20 0.43
GAA P10253 1/20 0.42
ALDH1A1 P00352 2/20 0.42
KDM4E B2RXH2 1/20 0.42
CNR1 P21554 1/20 0.42
CNR2 P34972 1/20 0.42
SPR P35270 1/20 0.42
EGLN1 Q9GZT9 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12516306 0.90 NPC1 (0.44) NPC1RAB9AMAPTSMN1; SMN2ALDH1A1
SCHEMBL2221780 0.81 KDM4E (0.47) KMT2AALDH1A1KDM4E
SCHEMBL29829548 0.79 BRS3 (0.38) KMT2AALDH1A1KDM4EEGLN1
SCHEMBL15746728 0.79 BRS3 (0.38) KMT2AALDH1A1KDM4EEGLN1
SCHEMBL1503149 0.79 KMT2A (0.48) NPC1RAB9AKMT2AMAPTSMN1; SMN2
SCHEMBL1503237 0.76 KMT2A (0.45) KMT2AMAPTGAAALDH1A1KDM4E
SCHEMBL1503172 0.76 KDM4E (0.45) NPC1RAB9AKMT2ASMN1; SMN2GAA
SCHEMBL27833103 0.75 KDM4E (0.46) KMT2AALDH1A1KDM4E
SCHEMBL22283906 0.75 KDM4E (0.37) KMT2AMAPTALDH1A1KDM4EEGLN1
SCHEMBL4306646 0.74 HCAR2 (0.35) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009146555-A1 HIV INTEGRASE INHIBITORS FROM PYRIDOXINE AMBRILIA BIOPHARMA INC. (CA) 2009-12-10 WO claimed