SCHEMBL4306646

SCHEMBL4306646

O=C(O)c1ncc(COCCc2ccc(F)cc2)c(CO)c1O

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.35
NR4A2 P43354 2/20 0.35
FFAR1 O14842 3/20 0.35
FFAR4 Q5NUL3 2/20 0.35
KDM5A P29375 1/20 0.35
KDM4C Q9H3R0 1/20 0.35
KDM5B Q9UGL1 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.33
XDH P47989 1/20 0.33
ALKBH1 Q13686 1/20 0.33
KMT2A Q03164 1/20 0.33
P4HTM Q9NXG6 1/20 0.33
BRS3 P32247 1/20 0.32
ME2 P23368 1/20 0.32
ME1 P48163 1/20 0.32
ME3 Q16798 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15746657 0.90 KDM4E (0.41) NR4A2KDM5AKDM4CKDM5BXDH
SCHEMBL1503195 0.89 HCAR2 (0.36) HCAR2FFAR1FFAR4KMT2A
SCHEMBL15746728 0.86 BRS3 (0.38) FFAR1KDM5AKDM4CKDM5BKMT2A
SCHEMBL29829548 0.86 BRS3 (0.38) FFAR1KDM5AKDM4CKDM5BKMT2A
SCHEMBL15746710 0.82 NR4A2 (0.45) NR4A2FFAR1FFAR4KDM4CALKBH1
SCHEMBL15746784 0.81 BCHE (0.37) KMT2A
SCHEMBL15746685 0.81 ALKBH1 (0.42) KDM5AKDM4CKDM5BALKBH1
SCHEMBL2221780 0.80 KDM4E (0.47) KMT2AP4HTM
SCHEMBL15746652 0.80 MAOB (0.38) KDM5AKDM4CKDM5B
SCHEMBL28791544 0.79 L3MBTL1 (0.42) HCAR2FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009146555-A1 HIV INTEGRASE INHIBITORS FROM PYRIDOXINE AMBRILIA BIOPHARMA INC. (CA) 2009-12-10 WO claimed
US-8742123-B2 HIV integrase inhibitors from pyridoxine TAIMED BIOLOGICS, INC. (TW) 2014-06-03 US disclosed