SCHEMBL4305262

SCHEMBL4305262

OC1CCOC(c2ccccn2)C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.38
ALDH1A1 P00352 2/20 0.38
MAPT P10636 2/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
KMT2A Q03164 1/20 0.38
KDM4E B2RXH2 1/20 0.37
PDE10A Q9Y233 1/20 0.36
JAK2 O60674 1/20 0.35
JAK1 P23458 1/20 0.35
JAK3 P52333 1/20 0.35
DDB1 Q16531 1/20 0.35
CRBN Q96SW2 1/20 0.35
LDHA P00338 1/20 0.34
GRM5 P41594 1/20 0.34
AXL P30530 1/20 0.34
FLT3 P36888 1/20 0.34
TYRO3 Q06418 1/20 0.34
MERTK Q12866 1/20 0.34
GAS6 Q14393 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31111388 0.84 HRH3 (0.43) HRH3ALDH1A1MAPTNPC1RAB9A
SCHEMBL31691890 0.76 HRH3 (0.43) HRH3ALDH1A1MAPTNPC1RAB9A
SCHEMBL8647354 0.76 HRH3 (0.43) HRH3ALDH1A1MAPTNPC1RAB9A
SCHEMBL1721948 0.76 PDE10A (0.43) ALDH1A1MAPTNPC1RAB9AKMT2A
SCHEMBL1721880 0.76 PDE10A (0.43) ALDH1A1MAPTNPC1RAB9AKMT2A
SCHEMBL1721946 0.76 PDE10A (0.43) ALDH1A1MAPTNPC1RAB9AKMT2A
SCHEMBL1721878 0.76 PDE10A (0.43) ALDH1A1MAPTNPC1RAB9AKMT2A
SCHEMBL1721879 0.76 PDE10A (0.43) ALDH1A1MAPTNPC1RAB9AKMT2A
SCHEMBL9156618 0.75 PIM1 (0.32) ALDH1A1KMT2A
SCHEMBL19819851 0.75 SLC6A3 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013010453-A1 CHEMOKING RECEPTOR ANTAGONISTS ABBOTT LABORATORIES (US) 2013-01-24 WO disclosed
WO-2009124882-A1 NOVEL PIPERIDINYL-1,3-DIHYDRO-BENZOIMIDAZOL-2-ONES AS M1 AGONISTS H. LUNDBECK A/S (DK) 2009-10-15 WO disclosed
WO-2009124882-A1 NOVEL PIPERIDINYL-1,3-DIHYDRO-BENZOIMIDAZOL-2-ONES AS M1 AGONISTS H. LUNDBECK A/S (DK) 2009-10-15 WO disclosed