SCHEMBL4307252

SCHEMBL4307252

[2H]C([2H])c1ccc(OCc2ccccc2)c([C@H](CC(=O)Cl)c2ccccc2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACP1 P24666 1/20 0.42
PTPN12 Q05209 1/20 0.42
PTPN13 Q12923 1/20 0.42
SSU72 Q9NP77 1/20 0.42
GLRA1 P23415 1/20 0.41
PTGER1 P34995 3/20 0.39
PTGER4 P35408 1/20 0.39
PTGER3 P43115 1/20 0.39
PTGER2 P43116 1/20 0.39
MRGPRX4 Q96LA9 2/20 0.39
FFAR4 Q5NUL3 1/20 0.39
KDM4E B2RXH2 1/20 0.38
LMNA P02545 1/20 0.38
ALDH1A1 P00352 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
KMT2A Q03164 2/20 0.38
NPC1 O15118 1/20 0.38
HPGD P15428 1/20 0.38
RAB9A P51151 1/20 0.38
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1990967 0.93 ACP1 (0.42) ACP1PTPN12PTPN13SSU72GLRA1
SCHEMBL1989523 0.92 PTGER1 (0.46) ACP1PTPN12PTPN13SSU72GLRA1
SCHEMBL1989522 0.92 PTGER1 (0.46) ACP1PTPN12PTPN13SSU72GLRA1
SCHEMBL1995519 0.85 KMT2A (0.45) ACP1PTPN12PTPN13SSU72PTGER1
SCHEMBL1990350 0.84 PTGER1 (0.51) PTGER1PTGER4PTGER3PTGER2MRGPRX4
SCHEMBL1990348 0.84 PTGER1 (0.51) PTGER1PTGER4PTGER3PTGER2MRGPRX4
SCHEMBL1992690 0.82 FOLH1 (0.42) ACP1PTPN12PTPN13SSU72GLRA1
SCHEMBL1992692 0.82 FOLH1 (0.42) ACP1PTPN12PTPN13SSU72GLRA1
SCHEMBL2167258 0.82 LRRK2 (0.46) PTGER1LMNAALDH1A1HPGDRAB9A
SCHEMBL15148415 0.82 LRRK2 (0.46) PTGER1LMNAALDH1A1HPGDRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009126844-A2 DERIVATIVES OF 3-(2-HYDROXY-5-METHYPHENYL)-N,N-DIISOPROPYL-3-PHENYLPROPYLAMINE AND METHODS OF USE THEREOF CONCERT PHARMACEUTICALS INC. (US) 2009-10-15 WO disclosed