SCHEMBL4313680

SCHEMBL4313680

Cn1c(=S)c2c(ncn2C)n(C)c1=S

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 8/20 0.52
ADORA2A P29274 3/20 0.52
POLB P06746 2/20 0.52
PIK3CD O00329 1/20 0.52
ADORA3 P0DMS8 1/20 0.52
CNR1 P21554 1/20 0.52
ACHE P22303 1/20 0.52
ADORA1 P30542 1/20 0.52
NTSR1 P30989 1/20 0.52
MC3R P41968 1/20 0.52
NOTUM Q6P988 1/20 0.52
SIRT3 Q9NTG7 1/20 0.52
GDA Q9Y2T3 1/20 0.52
NR2E1 Q9Y466 1/20 0.52
CYP3A4 P08684 2/20 0.44
PMP22 Q01453 2/20 0.44
MAPK1 P28482 1/20 0.44
BLM P54132 2/20 0.41
GLA P06280 1/20 0.41
PDE4A P27815 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9257690 0.81 ADORA2B (0.73) ADORA2BADORA2APOLBPIK3CDADORA3
Caffeine SCHEMBL8569482 0.68 ADORA2B (1.00) ADORA2BADORA2APOLBPIK3CDADORA3
Caffeine SCHEMBL10478364 0.68 ADORA2B (1.00) ADORA2BADORA2APOLBPIK3CDADORA3
Caffeine SCHEMBL5671 0.68 ADORA2B (1.00) ADORA2BADORA2APOLBPIK3CDADORA3
Caffeine SCHEMBL901194 0.68 ADORA2B (1.00) ADORA2BADORA2APOLBPIK3CDADORA3
SCHEMBL9644518 0.67 CYP3A4 (0.70) ADORA2BADORA2APOLBPIK3CDADORA3
Caffeine SCHEMBL23004680 0.67 ADORA2B (0.96) ADORA2BADORA2APOLBPIK3CDADORA3
Caffeine SCHEMBL569367 0.67 ADORA2B (0.96) ADORA2BADORA2APOLBPIK3CDADORA3
Caffeine SCHEMBL10407512 0.67 ADORA2B (0.96) ADORA2BADORA2APOLBPIK3CDADORA3
Caffeine SCHEMBL20637756 0.67 ADORA2B (0.96) ADORA2BADORA2APOLBPIK3CDADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7598019-B2 Method for cleavage of labile functional groups from chemical compounds UNIVERSITAT KONSTANZ (DE) 2009-10-06 US disclosed
US-20050255403-A1 Method for cleavage of labile functional groups from chemical compounds UNIVERSITAT KONSTANZ (DE) 2005-11-17 US disclosed
US-20050170281-A1 Method of cleaving labile functional groups from chemical compounds NIMBLEGEN SYSTEMS, INC. 2005-08-04 US disclosed
EP-1519941-A2 A METHOD OF CLEAVING LABILE FUNCTIONAL GROUPS FROM CHEMICAL COMPOUNDS Chemogenix GmbH (DE) 2005-04-06 EP disclosed
EP-1480927-A2 A METHOD FOR CLEAVAGE OF LABILE FUNCTIONAL GROUPS FROM CHEMICAL COMPOUNDS Universität Konstanz (DE) 2004-12-01 EP disclosed
WO-2004001033-A2 A METHOD OF CLEAVING LABILE FUNCTIONAL GROUPS FROM CHEMICAL COMPOUNDS CHEMOGENIX GMBH (DE) 2003-12-31 WO disclosed
WO-2003074542-A2 A METHOD FOR CLEAVAGE OF LABILE FUNCTIONAL GROUPS FROM CHEMICAL COMPOUNDS Universität Konstanz (DE) 2003-09-12 WO disclosed