SCHEMBL4314150

SCHEMBL4314150

CCc1ccc(C(N)=O)cc1.O=C(O)c1ccc2nc(-c3c(Cl)cccc3Cl)[nH]c2c1

nearest known ligand 0.60

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 16/20 0.60
DGAT1 O75907 2/20 0.53
ITGB1 P05556 1/20 0.50
ITGA4 P13612 1/20 0.50
ITGB7 P26010 1/20 0.50
HDAC3 O15379 1/20 0.50
HDAC1 Q13547 1/20 0.50
HDAC8 Q9BY41 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4314154 0.92 DGAT1 (0.53) CHEK2DGAT1ITGB1ITGA4ITGB7
SCHEMBL1248424 0.86 DGAT1 (0.67) CHEK2DGAT1ITGB1ITGA4ITGB7
SCHEMBL4011603 0.82 DGAT1 (0.57) CHEK2DGAT1HDAC3HDAC6
SCHEMBL1251104 0.82 DGAT1 (0.79) CHEK2DGAT1ITGB1ITGA4ITGB7
SCHEMBL1250981 0.80 DGAT1 (0.58) CHEK2DGAT1ITGB1ITGA4ITGB7
SCHEMBL3177289 0.78 NR4A2 (0.58) CHEK2DGAT1ITGB1ITGA4ITGB7
SCHEMBL3177891 0.78 DGAT1 (0.58) CHEK2DGAT1ITGB1ITGA4ITGB7
SCHEMBL1251886 0.77 DGAT1 (0.65) CHEK2DGAT1ITGB1ITGA4ITGB7
SCHEMBL1252157 0.77 DGAT1 (0.71) CHEK2DGAT1ITGB1ITGA4ITGB7
SCHEMBL3167498 0.76 DGAT1 (0.53) CHEK2DGAT1ITGB1ITGA4ITGB7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074089-A2 ORGANIC COMPOUNDS Novartis AG (CH) 2009-07-01 EP disclosed
WO-2008048991-A2 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2008-04-24 WO disclosed