SCHEMBL4314847

SCHEMBL4314847

C1CNCNC1.NC(=O)C1=CC=CC=CN1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5755219 0.85
SCHEMBL1117797 0.84 POLB (0.31)
Hydrochloric Acid SCHEMBL27832467 0.82 POLB (0.30)
Water SCHEMBL28206745 0.82 POLB (0.30)
Hydrogen Sulfide SCHEMBL28207789 0.82 POLB (0.30)
Hydrochloric Acid SCHEMBL28642702 0.82 POLB (0.30)
Hydrochloric Acid SCHEMBL28208398 0.81
Hydrochloric Acid SCHEMBL28207816 0.81
Trifluoroacetic Acid SCHEMBL28045656 0.73 L3MBTL1 (0.33)
SCHEMBL29575931 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090136570-A1 Taste-Masked Tablets and Granules UNIVERSITAT ZURICH (CH) 2009-05-28 US disclosed
WO-2007087188-A2 TASTE-MASKED TABLETS AND GRANULES MERCK & CO., INC. (US) 2007-08-02 WO disclosed
WO-2006060225-A2 PROCESS FOR ASYMMETRIC SYNTHESIS OF HEXAHYDROPYRIMIDO[1,2-A] AZEPINE-2-CARBOXAMIDES AND RELATED COMPOUNDS MERCK & CO., INC. (US) 2006-06-08 WO disclosed