SCHEMBL4318906

SCHEMBL4318906

COc1ncnc2[nH]cc(C(O)c3c(F)ccc(N)c3F)c12

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 5/20 0.42
CYP2C19 P33261 3/20 0.40
CYP3A4 P08684 3/20 0.39
TRPA1 O75762 4/20 0.36
LRRK2 Q5S007 4/20 0.33
MAP3K7 O43318 3/20 0.32
TAB1 Q15750 3/20 0.32
BTK Q06187 1/20 0.32
JAK3 P52333 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4318902 0.85 CYP2C9 (0.45) CYP2C9CYP2C19CYP3A4TRPA1MAP3K7
SCHEMBL4324611 0.85 CYP3A4 (0.39) CYP2C9CYP2C19CYP3A4TRPA1LRRK2
SCHEMBL1086260 0.79 CYP2C9 (0.54) CYP2C9CYP2C19CYP3A4
SCHEMBL3709081 0.77 CDK2 (0.43) CYP3A4TRPA1LRRK2
SCHEMBL3505507 0.76 MTNR1A (0.38) CYP2C9CYP3A4
SCHEMBL3700075 0.74 CDC7 (0.34) CYP3A4
SCHEMBL1086078 0.73 CYP2C9 (0.65) CYP2C9CYP2C19CYP3A4
SCHEMBL3701118 0.72 GRM8 (0.40) LRRK2JAK3
SCHEMBL3505627 0.72 BRAF (0.41) CYP2C9CYP2C19CYP3A4BTK
SCHEMBL1816955 0.72 CYP2C9 (0.37) CYP2C9CYP2C19CYP3A4JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009143024-A2 COMPOUNDS AND METHODS FOR KINASE MODULATION, AND INDICATIONS THEREFOR PLEXXIKON, INC. (US) 2009-11-26 WO disclosed