SCHEMBL4320462

SCHEMBL4320462

O=c1[nH]c(=O)c2[nH]c(CCCc3cnn(Cc4ccc(F)c(F)c4)c3)nc2[nH]1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 8/20 0.41
ADORA1 P30542 4/20 0.41
ADORA2A P29274 3/20 0.41
SCD O00767 1/20 0.37
KLKB1 P03952 1/20 0.36
ALK Q9UM73 1/20 0.35
ADORA3 P0DMS8 4/20 0.35
HDAC1 Q13547 1/20 0.34
CLPP Q16740 1/20 0.33
SCD5 Q86SK9 1/20 0.33
DAO P14920 1/20 0.32
P2RX7 Q99572 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4013561 0.81 ADORA2B (0.42) ADORA2BADORA1ADORA2AADORA3
SCHEMBL5685358 0.78 ADORA2B (0.45) ADORA2BADORA1ADORA2AADORA3
SCHEMBL5685510 0.76 ADORA2B (0.49) ADORA2BADORA1ADORA2ASCDADORA3
SCHEMBL5608377 0.73 ADORA2B (0.50) ADORA2BADORA1ADORA2AADORA3
SCHEMBL1720832 0.69 ADORA2B (0.37) ADORA2BDAO
SCHEMBL2822621 0.66 ALK (0.45) ADORA2BADORA1ADORA2ASCDKLKB1
SCHEMBL1065674 0.66 ADORA2B (0.62) ADORA2BADORA1ADORA2AADORA3
SCHEMBL15642930 0.65 HCAR2 (0.43) ADORA2BADORA1ADORA2AADORA3HDAC1
Hydrochloric Acid SCHEMBL21492821 0.65 MAPT (0.48) ADORA2BADORA1ADORA2ASCDKLKB1
SCHEMBL30012217 0.64 ADORA2B (0.71) ADORA2BADORA1ADORA2AADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009088518-A1 A2B ADENOSINE RECEPTOR ANTAGONISTS FOR THE TREATMENT OF CANCER CV THERAPEUTICS, INC. (US) 2009-07-16 WO disclosed
EP-1622908-A1 XANTHINE DERIVATIVES AS A2B ADENOSINE RECEPTOR ANTAGONISTS CV THERAPEUTICS, INC. (US) 2006-02-08 EP disclosed
WO-2004106337-A1 XANTHINE DERIVATIVES AS A2B ADENOSINE RECEPTOR ANTAGONISTS CV THERAPEUTICS, INC. (US) 2004-12-09 WO disclosed