SCHEMBL4320736

SCHEMBL4320736

COCCc1cc(Cl)c(Cl)c(CN(C(=O)O)C2CC2)c1

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
REN P00797 19/20 0.56
KCNH2 Q12809 9/20 0.56
SLC6A2 P23975 1/20 0.44
SLC6A4 P31645 1/20 0.44
SLC6A3 Q01959 1/20 0.44
CYP3A4 P08684 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1080226 0.85 REN (0.51) RENKCNH2SLC6A2SLC6A4SLC6A3
SCHEMBL4315675 0.84 REN (0.45) RENKCNH2SLC6A2SLC6A4SLC6A3
SCHEMBL1073880 0.84 REN (0.49) RENKCNH2SLC6A2SLC6A4SLC6A3
SCHEMBL663545 0.81 REN (0.47) RENKCNH2CYP3A4
SCHEMBL663478 0.78 SLC6A4 (0.41) RENKCNH2SLC6A2SLC6A4SLC6A3
SCHEMBL13625719 0.78 REN (0.60) RENKCNH2CYP3A4
SCHEMBL663581 0.76 SLC6A4 (0.44) RENKCNH2SLC6A2SLC6A4SLC6A3
SCHEMBL1072075 0.76 REN (0.54) RENKCNH2CYP3A4
SCHEMBL4686564 0.74 REN (0.48) RENKCNH2CYP3A4
SCHEMBL4686561 0.74 REN (0.48) RENKCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009140769-A1 3, 4 - SUBSTITUTED PIPERIDINE DERIVATIVES AS RENIN INHIBITORS MERCK FROSST CANADA LTD. (CA) 2009-11-26 WO disclosed