SCHEMBL4322993

SCHEMBL4322993

CN(Cc1ccc(OC(F)(F)F)cc1)C(=O)C1c2ccccc2C(=O)N1C1CN(C(=O)O)C1

nearest known ligand 0.58

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 20/20 0.58
SCN5A Q14524 11/20 0.58
KCNH2 Q12809 11/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4323000 0.82 SCN9A (0.80) SCN9ASCN5AKCNH2
SCHEMBL4329573 0.75 SCN9A (0.66) SCN9ASCN5AKCNH2
SCHEMBL4322988 0.75 SCN9A (0.64) SCN9ASCN5AKCNH2
SCHEMBL4326444 0.74 SCN9A (0.80) SCN9ASCN5AKCNH2
SCHEMBL13577840 0.73 SCN9A (1.00) SCN9ASCN5AKCNH2
SCHEMBL4318437 0.73 SCN9A (0.76) SCN9ASCN5AKCNH2
SCHEMBL4323513 0.73 SCN9A (0.81) SCN9ASCN5AKCNH2
SCHEMBL4325794 0.72 SCN9A (0.63) SCN9ASCN5AKCNH2
SCHEMBL4329960 0.71 SCN9A (0.73) SCN9ASCN5AKCNH2
SCHEMBL4334944 0.71 SCN9A (0.43) SCN9ASCN5AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009145721-A1 ISOINDOLINE DERIVATIVES COMPRISING PHENYL GROUPS AND THEIR USE IN THE TREATMENT OF PAIN DISORDERS ASTRAZENECA AB (SE) 2009-12-03 WO claimed
WO-2009145721-A1 ISOINDOLINE DERIVATIVES COMPRISING PHENYL GROUPS AND THEIR USE IN THE TREATMENT OF PAIN DISORDERS ASTRAZENECA AB (SE) 2009-12-03 WO disclosed