SCHEMBL43231

SCHEMBL43231

O=C(CBr)NCCC(=O)ON1C(=O)CCC1=O

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HDAC3 O15379 2/20 0.33
HDAC4 P56524 2/20 0.33
HDAC1 Q13547 2/20 0.33
HDAC7 Q8WUI4 2/20 0.33
HDAC2 Q92769 2/20 0.33
HDAC10 Q969S8 2/20 0.33
HDAC11 Q96DB2 2/20 0.33
HDAC8 Q9BY41 2/20 0.33
HDAC6 Q9UBN7 2/20 0.33
HDAC9 Q9UKV0 2/20 0.33
HDAC5 Q9UQL6 2/20 0.33
AANAT Q16613 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20091594 0.94 HPGD (0.33) HPGDHTTSMN1; SMN2HDAC3HDAC4
SCHEMBL8735537 0.91 HPGD (0.37) HPGDHTTSMN1; SMN2HDAC3HDAC4
SCHEMBL13001926 0.90 HPGD (0.33) HPGDHTTSMN1; SMN2
SCHEMBL3705350 0.88 HDAC3 (0.44) HPGDHTTSMN1; SMN2HDAC3HDAC4
SCHEMBL16453924 0.87 HPGD (0.38) HPGDHTTSMN1; SMN2
SCHEMBL24045358 0.87 HPGD (0.31) HPGDHTTSMN1; SMN2
SCHEMBL20091644 0.86 HPGD (0.34) HPGDHTTSMN1; SMN2
SCHEMBL1577786 0.86 SMN1; SMN2 (0.37) HPGDHTTSMN1; SMN2
SCHEMBL11913384 0.86 SMN1; SMN2 (0.37) HPGDHTTSMN1; SMN2
SCHEMBL15669350 0.86 SMN1; SMN2 (0.37) HPGDHTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 4322 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025235971-A1 METHODS FOR DETECTING DNA SEQUENCE VARIATION IN THICK TISSUE SECTIONS THE JOHNS HOPKINS UNIVERSITY (US) 2025-11-13 WO claimed
US-20250295745-A1 CROSS-LINKED TUMOR LYSATE SPHERICAL NUCLEIC ACIDS AS CANCER VACCINES NORTHWESTERN UNIVERSITY 2025-09-25 US claimed
EP-4615969-A1 METHODS FOR DETECTING RNA AND MOLECULAR ANALYSIS IN THICK TISSUE SECTIONS The Johns Hopkins University (US) 2025-09-17 EP claimed
CN-112533640-B Targeting of M2-type tumor-associated macrophages using melittin-based apoptosis-inducing peptides 双亥生命科学株式会社 2025-02-28 CN claimed
US-12070543-B2 Blood processing apparatus and method for detoxifying bacterial lipopolysaccharide in vivo ORTH CONSULTING, LLC (US) 2024-08-27 US claimed
WO-2024103007-A1 METHODS FOR DETECTING RNA AND MOLECULAR ANALYSIS IN THICK TISSUE SECTIONS THE JOHNS HOPKINS UNIVERSITY (US) 2024-05-16 WO claimed
US-20230414855-A1 Blood Processing Apparatus and Method for Detoxifying Bacterial Lipopolysaccharide In Vivo ORTH CONSULTING, LLC 2023-12-28 US claimed
EP-3362089-B1 IMMUNOGENIC COMPOSITIONS AGAINST S. AUREUS SANOFI PASTEUR (FR) 2023-12-06 EP claimed
WO-2023220678-A1 CROSS-LINKED TUMOR LYSATE SPHERICAL NUCLEIC ACIDS AS CANCER VACCINES NORTHWESTERN UNIVERSITY (US) 2023-11-16 WO claimed
US-11725222-B2 Cleavable nucleotide analogs and uses thereof PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2023-08-15 US claimed
WO-2007120579-A2 LOADED LATEX OPTICAL MOLECULAR IMAGING PROBES CARESTREAM HEALTH, INC. (US) 2007-10-25 WO claimed
WO-2007046865-A1 BIOLOGICAL INDICATOR STERIS, INC. (US) 2007-04-26 WO claimed
EP-1776389-A2 SIALIC ACID DERIVATIVES Lipoxen Technologies Limited (GB) 2007-04-25 EP claimed
US-20060269983-A1 Biological indicator AMERICAN STERILIZER COMPANY 2006-11-30 US claimed
WO-2006090119-A1 ACTIVATED SIALIC ACID DERIVATIVES FOR PROTEIN DERIVATISATION AND CONJUGATION LIPOXEN TECHNOLOGIES LIMITED (GB) 2006-08-31 WO claimed
EP-1689846-A2 METHOD OF TARGETING SPECIFIC CELL POPULATIONS USING CELL-BINDING AGENT MAYTANSINOID CONJUGATES LINKED VIA A NON-CLEAVABLE LINKER, SAID CONJUGATES, AND METHODS OF MAKING SAID CONJUGATES Immunogen, Inc. (US) 2006-08-16 EP claimed
WO-2006016168-A2 SIALIC ACID DERIVATIVES LIPOXEN TECHNOLOGIES LIMITED (GB) 2006-02-16 WO claimed
US-20050169933-A1 Method of targeting specific cell populations using cell-binding agent maytansinoid conjugates linked via a non-cleavable linker, said conjugates, and methods of making said conjugates IMMUNOGEN, INC. 2005-08-04 US claimed
WO-2005037992-A2 METHOD OF TARGETING SPECIFIC CELL POPULATIONS USING CELL-BINDING AGENT MAYTANSINOID CONJUGATES LINKED VIA A NON-CLEAVABLE LINKER, SAID CONJUGATES, AND METHODS OF MAKING SAID CONJUGATES IMMUNOGEN, INC. (US) 2005-04-28 WO claimed
WO-2004089295-A2 HOMOGENEOUS AND HETEROGENEOUS ASSAY METHODS USING NUCLEATION CENTERS AND NOVEL COVALENT CHEMISTRIES FOR THE RAPID MEASUREMENT OF PHOSPHORYLATION AND DE-PHOSPHORYLATION CHROMAGEN, INC. (US) 2004-10-21 WO claimed