SCHEMBL4326786

SCHEMBL4326786

O=C(O)Nc1ccccc1N1CCOCC1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.70
CYP1A2 P05177 1/20 0.70
CYP3A4 P08684 1/20 0.70
CYP2C19 P33261 1/20 0.70
KMT2A Q03164 2/20 0.64
MEN1 O00255 1/20 0.64
L3MBTL1 Q9Y468 1/20 0.64
POLB P06746 3/20 0.64
SCN9A Q15858 1/20 0.64
SMN1; SMN2 Q16637 4/20 0.62
KCNQ2 O43526 1/20 0.62
PKM P14618 1/20 0.62
TDP1 Q9NUW8 1/20 0.62
TSHR P16473 3/20 0.61
EPHX2 P34913 1/20 0.61
HPGD P15428 1/20 0.61
MAPK10 P53779 1/20 0.61
HTT P42858 1/20 0.61
ATM Q13315 1/20 0.60
MCOLN3 Q8TDD5 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20910885 0.89 ALDH1A1 (0.68) ALDH1A1CYP1A2CYP3A4CYP2C19KMT2A
SCHEMBL9555514 0.86 POLB (0.69) ALDH1A1CYP1A2CYP3A4CYP2C19KMT2A
SCHEMBL20911012 0.85 ALDH1A1 (0.64) ALDH1A1CYP1A2CYP3A4CYP2C19KMT2A
SCHEMBL4318899 0.85 KCNQ2 (0.68) ALDH1A1CYP1A2CYP3A4KMT2AMEN1
SCHEMBL328566 0.84 ALDH1A1 (0.70) ALDH1A1CYP1A2CYP3A4CYP2C19KMT2A
SCHEMBL4717225 0.82 ALDH1A1 (0.60) ALDH1A1CYP1A2CYP3A4CYP2C19KMT2A
SCHEMBL5903997 0.82 ALDH1A1 (0.71) ALDH1A1CYP1A2CYP3A4CYP2C19KMT2A
SCHEMBL19889013 0.82 ALDH1A1 (0.60) ALDH1A1CYP1A2CYP3A4CYP2C19KMT2A
SCHEMBL18701666 0.82 ALDH1A1 (0.62) ALDH1A1CYP1A2CYP3A4CYP2C19KMT2A
SCHEMBL18711850 0.82 ALDH1A1 (0.70) ALDH1A1CYP1A2CYP3A4CYP2C19KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009090548-A2 3-AZABICYCLO [3.1.0] HEXANE DERIVATIVES AS VANILLOID RECEPTOR LIGANDS GLENMARK PHARMACEUTICALS, S.A. (US) 2009-07-23 WO disclosed
EP-0525197-B1 3-BENZYLIDENE-1-CARBAMOYL-2-PYRROLIDONE ANALOGS SHIONOGI & CO (JP) 1997-08-27 EP disclosed
US-5319100-A Antiinflammatory agent which does not cause stomach diseases SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1994-06-07 US disclosed
US-5319099-A Antiinflammatory agent which does not cause stomach diseases SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1994-06-07 US disclosed
EP-0525197-A1 3-BENZYLIDENE-1-CARBAMOYL-2-PYRROLIDONE ANALOG SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1993-02-03 EP disclosed