SCHEMBL4334787

SCHEMBL4334787

Cc1cc(OCc2ccc(F)c(F)c2)cc(C)c1N

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAOB P27338 11/20 0.52
MAOA P21397 2/20 0.52
ACHE P22303 1/20 0.48
ANO1 Q5XXA6 1/20 0.40
HTR6 P50406 2/20 0.40
PPARA Q07869 1/20 0.39
NOS1 P29475 1/20 0.39
NOS2 P35228 1/20 0.39
FFAR1 O14842 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1578198 0.84 MAOB (0.43) MAOBMAOAACHEANO1
SCHEMBL1578651 0.83 MAOB (0.59) MAOBMAOAACHE
SCHEMBL4323959 0.80 MAOB (0.54) MAOBMAOAACHE
SCHEMBL4322263 0.80 MAOB (0.53) MAOBMAOAACHE
SCHEMBL4319284 0.79 MAOB (0.65) MAOBMAOAACHE
SCHEMBL5382147 0.78 MAOB (0.66) MAOBMAOA
SCHEMBL1578355 0.78 MAOB (0.50) MAOBMAOAACHEANO1PPARA
SCHEMBL25947183 0.77 MAOB (0.50) MAOB
SCHEMBL4323948 0.77 MAOB (0.53) MAOBMAOA
SCHEMBL25947185 0.77 MAOB (0.57) MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8492588-B2 Benzyloxy anilide derivatives useful as potassium channel modulators VALEANT PHARMACEUTICALS INTERNATIONAL (US) 2013-07-23 US disclosed
US-20120329869-A1 BENZYLOXY ANILIDE DERIVATIVES USEFUL AS POTASSIUM CHANNEL MODULATORS VALEANT PHARMACEUTICALS INTERNATIONAL 2012-12-27 US disclosed
US-8188314-B2 Benzyloxy anilide derivatives useful as potassium channel modulators VALEANT PHARMACEUTICALS INTERNATIONAL (US) 2012-05-29 US disclosed
US-20090326059-A1 BENZYLOXY ANILIDE DERIVATIVES USEFUL AS POTASSIUM CHANNEL MODULATORS VALEANT PHARMACEUTICALS INTERNATIONAL (US) 2009-12-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120329869-A1 BENZYLOXY ANILIDE DERIVATIVES USEFUL AS POTASSIUM CHANNEL MODULATORS KCND2, KCNB2, KCNAB1 MAOB 549/4885MAOA 756/4885ACHE 1604/4885
US-20090326059-A1 BENZYLOXY ANILIDE DERIVATIVES USEFUL AS POTASSIUM CHANNEL MODULATORS KCND2, KCNB2, KCNAB1 MAOB 549/4885MAOA 756/4885ACHE 1604/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.