SCHEMBL4334916

SCHEMBL4334916

CC(C)(C)OC(=O)C1=CC=CNN=C1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32
CA14 Q9ULX7 1/20 0.32
GABRA1 P14867 2/20 0.32
GABRG2 P18507 2/20 0.32
GABRB3 P28472 2/20 0.32
GABRA5 P31644 2/20 0.32
GABRA3 P34903 2/20 0.32
GABRA2 P47869 2/20 0.32
ALDH1A1 P00352 3/20 0.31
TSHR P16473 1/20 0.31
HSD17B10 Q99714 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
ABCG2 Q9UNQ0 1/20 0.30
LMNA P02545 1/20 0.30
GABRP O00591 1/20 0.30
GABRD O14764 1/20 0.30
GABRB1 P18505 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28296128 0.81 TSHR (0.35) CA12CA1CA2CA9CA14
SCHEMBL25195357 0.75 CA12 (0.34) CA12CA1CA2CA9CA14
SCHEMBL28379616 0.74 TP53 (0.32) GABRA1GABRG2GABRB3GABRA5GABRA3
Hydrochloric Acid SCHEMBL27029865 0.73 CA12 (0.33) CA12CA1CA2CA9CA14
SCHEMBL30356678 0.72 TP53 (0.33) HSD17B10
SCHEMBL28379615 0.66 TP53 (0.33) HSD17B10
SCHEMBL4334920 0.65 ALDH1A1 (0.30) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL10512179 0.65 TP53 (0.31) CA12CA1CA2CA9CA14
SCHEMBL6619765 0.63 ALDH1A1 (0.33) CA12CA1CA2CA9CA14
SCHEMBL29152579 0.63 TP53 (0.33) CA12CA1CA2CA9CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106061944-A Pyridines and pyrimidines and use thereof 普渡制药公司 2016-10-26 CN claimed
CN-117412959-A Substituted 1-aryl-1 '-heteroaryl compounds, substituted 1,1' -biaryl compounds, and methods of use thereof 爱彼特生物制药公司 2024-01-16 CN disclosed
CN-106061944-A Pyridines and pyrimidines and use thereof 普渡制药公司 2016-10-26 CN disclosed
WO-2009145357-A1 IN 1-POSITION DURCH EINEN RING SUBSTITUIERTE BENZO [1, 4] DIAZEPINE ZUR VERWENDUNGS ALS ANTIDEPRESSIVA OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2009-12-03 WO disclosed