SCHEMBL434563

SCHEMBL434563

COC(=O)c1ccc2c(c1)CC(NC(=O)C1(C)CCN(C(=O)O)CC1)CC2

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 2/20 0.43
MTNR1B P49286 2/20 0.43
CA1 P00915 3/20 0.41
CA2 P00918 3/20 0.41
ACHE P22303 3/20 0.41
OPRD1 P41143 1/20 0.39
HDAC8 Q9BY41 5/20 0.37
CNR2 P34972 1/20 0.36
DRD4 P21917 1/20 0.36
KDM5A P29375 3/20 0.36
KDM4E B2RXH2 1/20 0.36
NPC1 O15118 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
RAB9A P51151 1/20 0.36
HDAC6 Q9UBN7 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL354658 0.89 NPC1 (0.42) MTNR1AMTNR1BCA1CA2ACHE
SCHEMBL355075 0.82 MTNR1A (0.39) MTNR1AMTNR1BCA1CA2ACHE
SCHEMBL355074 0.80 MTNR1A (0.38) MTNR1AMTNR1BCA1CA2ACHE
SCHEMBL354456 0.78 HDAC8 (0.46) HDAC8HDAC6
SCHEMBL469781 0.74 MTNR1A (0.51) MTNR1AMTNR1BCA1CA2ACHE
SCHEMBL354927 0.74 MTNR1A (0.52) MTNR1AMTNR1BCA1CA2ACHE
SCHEMBL464149 0.73 MTNR1A (0.50) MTNR1AMTNR1BCA1CA2ACHE
SCHEMBL10253259 0.73 MTNR1A (0.51) MTNR1AMTNR1BCA1CA2ACHE
SCHEMBL354268 0.73 MTNR1A (0.51) MTNR1AMTNR1BCA1CA2ACHE
SCHEMBL355482 0.72 EPHX2 (0.53) MTNR1AMTNR1BCA1CA2ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012012322-A1 SUBSTITUTED HYDROXAMIC ACIDS AND USES THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2012-01-26 WO disclosed