SCHEMBL4346800

SCHEMBL4346800

OCc1cc(NCc2ccccc2Sc2cccc(Cl)c2)ccc1O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 2/20 0.48
SLC6A2 P23975 1/20 0.48
SLC6A3 Q01959 1/20 0.48
EGFR P00533 2/20 0.41
NOX4 Q9NPH5 2/20 0.40
MAPT P10636 4/20 0.40
HPGD P15428 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
MAOB P27338 2/20 0.37
PLA2G1B P04054 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12846506 0.88 SMN1; SMN2 (0.51) EGFRNOX4MAPTHPGDSMN1; SMN2
SCHEMBL4345369 0.88 SLC6A4 (0.44) SLC6A4EGFRNOX4MAPTHPGD
SCHEMBL4345562 0.88 SLC6A2 (0.50) SLC6A4SLC6A2SLC6A3EGFRNOX4
SCHEMBL4356200 0.88 NOX4 (0.48) EGFRNOX4MAPTHPGDSMN1; SMN2
SCHEMBL4346742 0.86 MAPT (0.45) EGFRNOX4MAPTHPGDSMN1; SMN2
SCHEMBL4354072 0.86 SLC6A2 (0.48) SLC6A4SLC6A2SLC6A3EGFRNOX4
SCHEMBL4355493 0.84 NOX4 (0.60) SLC6A4SLC6A2SLC6A3EGFRNOX4
SCHEMBL4346454 0.83 NOX4 (0.43) SLC6A4EGFRNOX4MAPTHPGD
SCHEMBL4341606 0.82 SLC6A4 (0.51) SLC6A4SLC6A2SLC6A3SMN1; SMN2CA12
SCHEMBL4345796 0.82 EGFR (0.53) SLC6A4SLC6A2SLC6A3EGFRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-1539683-A2 PHENOL DERIVATIVES AND THEIR USE AS ROTAMASE INHIBITORS Jerini AG (DE) 2005-06-15 EP claimed
WO-2004030664-A2 NEW COMPOUNDS FOR THE INHIBITION OF UNDESIRED CELL PROLIFERATION AND USE THEREOF JERINI AG (DE) 2004-04-15 WO claimed
WO-2004026815-A2 PHENOL DERIVATIVES AND THEIR USE AS ROTAMASE INHIBITORS JERINI AG (DE) 2004-04-01 WO claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed