SCHEMBL4347124

SCHEMBL4347124

O=C(NCCc1ccccc1)Nc1cc(Cl)c(O)c(-c2nc3ccccc3s2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.48
MAPT P10636 9/20 0.47
RAB9A P51151 3/20 0.47
NPC1 O15118 2/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
CNR1 P21554 1/20 0.47
KDM4E B2RXH2 2/20 0.46
NAMPT P43490 3/20 0.46
THRB P10828 1/20 0.46
RXFP1 Q9HBX9 2/20 0.45
CTSD P07339 1/20 0.44
MGLL Q99685 1/20 0.44
PRMT3 O60678 1/20 0.43
MAOB P27338 1/20 0.43
SNCA P37840 1/20 0.43
TP53 P04637 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
EPHX1 P07099 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4344552 0.90 NAMPT (0.57) EPHX2MAPTRAB9ANPC1MEN1
SCHEMBL4348632 0.86 CSNK1D (0.53) MAPTRAB9ANPC1MEN1KMT2A
SCHEMBL6519124 0.83 MAPT (0.47) MAPTRAB9ANPC1SMN1; SMN2KDM4E
SCHEMBL4561504 0.80 MAPT (0.54) MAPTRAB9ANPC1MEN1KMT2A
SCHEMBL4352804 0.80 MAPT (0.56) MAPTRAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL4351106 0.80 CNR1 (0.68) MAPTRAB9ANPC1MEN1KMT2A
SCHEMBL6251830 0.79 NAMPT (0.37) EPHX2MAPTRAB9ANPC1MEN1
SCHEMBL4341723 0.78 MAPT (0.49) MAPTRAB9ANPC1MEN1KMT2A
SCHEMBL4354538 0.78 SMN1; SMN2 (0.52) MAPTRAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL4355895 0.77 RAB9A (0.58) EPHX2MAPTRAB9ANPC1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed