SCHEMBL4347138

SCHEMBL4347138

O=C(Nc1ccc(OC(F)(F)F)cc1)Nc1ccc(O)c(F)c1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 8/20 0.71
FAAH O00519 1/20 0.57
MAPT P10636 2/20 0.56
MEN1 O00255 1/20 0.56
TP53 P04637 1/20 0.56
CASP3 P42574 1/20 0.56
HTT P42858 1/20 0.56
KMT2A Q03164 1/20 0.56
NPSR1 Q6W5P4 1/20 0.56
SENP7 Q9BQF6 1/20 0.56
NPC1 O15118 1/20 0.54
RAB9A P51151 1/20 0.54
EPHX1 P07099 2/20 0.51
BRAF P15056 1/20 0.51
KDR P35968 1/20 0.51
IDH1 O75874 2/20 0.50
HDAC3 O15379 1/20 0.50
HDAC4 P56524 1/20 0.50
HDAC1 Q13547 1/20 0.50
HDAC7 Q8WUI4 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4349998 0.87 EPHX2 (0.73) EPHX2FAAHMAPTMEN1TP53
SCHEMBL11555827 0.84 EPHX2 (1.00) EPHX2FAAHMAPTMEN1TP53
SCHEMBL4343951 0.84 EPHX2 (0.69) EPHX2FAAHMAPTMEN1TP53
SCHEMBL4106154 0.84 EPHX2 (0.69) EPHX2FAAHMAPTMEN1TP53
SCHEMBL12217997 0.82 EPHX2 (0.86) EPHX2FAAHMAPTMEN1TP53
SCHEMBL18031167 0.82 EPHX2 (0.86) EPHX2FAAHMAPTMEN1TP53
SCHEMBL4351078 0.80 MEN1 (0.67) EPHX2FAAHMAPTMEN1TP53
SCHEMBL4352985 0.80 CA12 (0.58) FAAHMAPTMEN1KMT2ANPSR1
SCHEMBL26154100 0.80 EPHX2 (0.71) EPHX2FAAHMAPTMEN1TP53
SCHEMBL6229951 0.79 CA12 (0.60) FAAHMAPTMEN1TP53HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100546977-C Suppress the new compound and the application thereof of rotamase JERINI AG (DE) 2009-10-07 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed